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2-{3-oxo-9-[(1R,2R)-2-phenylcyclopropanecarbonyl]-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
4-(4-phenyl-1H-pyrazol-5-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
5-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindole-2-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-(azocan-1-yl)-3-[2-methoxy-4-(1,2-oxazinan-2-ylmethyl)phenoxy]propan-2-ol
1-(4-ethylpiperazin-1-yl)-3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propan-1-one
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3-(1H-indol-3-yl)propanamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]benzamide
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]acetamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-methoxypropanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-[(1H-indol-5-ylmethyl)amino]-4-methylpyrimidin-5-yl}ethan-1-one
(2R,3S,6R)-3-(4-fluorophenyl)-5-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2,3-dihydro-1H-inden-1-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
2-(2-{1-[3-(dimethylamino)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
3-(azocan-1-yl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]propanamide
methyl 2-{3-[({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]-1H-indol-1-yl}acetate
4-(2H-1,3-benzodioxol-5-ylmethyl)-N-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-3-oxopiperazine-1-carboxamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-cyclopentanecarbonylpiperidine-4-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-3-{5-[(4-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
2-(2-methoxyethyl)-8-(5-propyl-1,2-oxazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(3-methoxyphenyl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1,2,4-triazin-3-amine
(4aR,8aS)-1-butyl-6-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
3-{[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]methyl}-8-methyl-1,2-dihydroquinolin-2-one
1-{4-[(ethylamino)methyl]-2-methoxyphenoxy}-3-(morpholin-4-yl)propan-2-ol
N-cyclopropyl-1,3-dimethyl-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}-1H-pyrazole-5-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
N-[2-(dimethylamino)ethyl]-3-methyl-N-[(5-methylthiophen-2-yl)methyl]-4-oxo-3,4-dihydrophthalazine-1-carboxamide
5-[5-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)thiophen-2-yl]-1H-pyrazole
3-[4-(6-carbamoylpyrazin-2-yl)phenyl]propanoic acid
methyl 3-(4-tert-butylbenzenesulfonamidomethyl)-5-(pyrazine-2-amido)benzoate
N-[1-(1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}piperidin-4-yl)-2-phenylethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
(3aR,6aR)-2-cyclopentyl-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[(4-fluorophenyl)methyl]-2,6-dimethyl-N-(oxolan-2-ylmethyl)pyrimidine-4-carboxamide
8-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(1,2-benzoxazol-3-yl)-N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}acetamide
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-methylazepane-2-carboxamide
2-tert-butyl-4-hydroxy-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}pyrimidine-5-carboxamide
1-[(2-methoxyphenyl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
(4aS,7aR)-1-[(4-fluorophenyl)methyl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-(4-methanesulfonylphenyl)-1H-pyrazol-1-yl]propanoic acid
4-(5-propyl-1,2-oxazole-3-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-[2-(2-methyl-1H-imidazol-1-yl)acetyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
8-{[4-(2,2-dimethylmorpholine-4-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
2-[3-(2,6-difluorophenyl)-1H-pyrazol-1-yl]-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
4-[3-(1-methyl-1H-imidazole-2-carbonyl)phenyl]-6-(1H-pyrazol-1-yl)pyrimidine
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-3-carboxamide
(3S,4R)-1-(1H-indole-5-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
6-(4-fluoro-2-methoxyphenyl)-N2-(4-methylphenyl)-1,3,5-triazine-2,4-diamine
2-methyl-7-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
1-(4-{[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one