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(2-{[4-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-1-yl]methyl}phenyl)methanol
4-(1H-imidazol-1-yl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-4-carboxylic acid
2-methyl-N-(2-{pyrazolo[1,5-a]pyridin-7-yl}pyridin-3-yl)propanamide
1-[3-(3-hydroxy-3-methylbutyl)benzoyl]-4-phenylpiperidine-4-carbonitrile
1-[2-(methylsulfanyl)pyrimidin-4-yl]-N-[2-(pyridin-3-yl)ethyl]piperidin-4-amine
N-(5-hydroxyadamantan-2-yl)-7-(2-methoxyacetamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
methyl 4-({[5-(3-methoxyphenyl)-1,2,4-triazin-3-yl]amino}methyl)benzoate
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-3-[2-(4-fluorophenyl)ethyl]piperidine
2-[(cyclopropylmethyl)sulfanyl]-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
(3S,5S)-1-[(3-fluoro-2-methylphenyl)methyl]-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2-(dimethylamino)-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-2-(3-methylphenyl)acetamide
2-[methyl({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl})amino]ethan-1-ol
(4aS,8aR)-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
(3S,9aR)-8-(3,5-dichlorobenzoyl)-3-[(1R)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
ethyl 2-(2-{2-[(3,5-dimethylphenyl)carbamoyl]acetamido}ethyl)-1,3-thiazole-4-carboxylate
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(dimethylamino)ethan-1-one
N-[(2,4-dimethoxyphenyl)methyl]-1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
1-[(2-aminopyridin-3-yl)methyl]-4-(4-fluoro-2-methylphenoxy)piperidine-4-carboxylic acid
1-(1-methyl-1H-pyrazole-4-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[methyl(phenyl)amino]ethan-1-one
2-methyl-2-[4-(morpholin-4-yl)-2-({[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}amino)pyrimidin-5-yl]propanoic acid
propan-2-yl 4-(4-methoxyphenyl)-2-methyl-3-oxopiperazine-1-carboxylate
ethyl 1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
4-{1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1H-imidazol-2-yl}quinoline
7-methyl-3-[2-(1-methylpiperidin-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
3,5-dimethyl-4-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-2-yl]-1,2-oxazole
3-{2-[(2-chlorophenyl)methyl]morpholine-4-carbonyl}-1-methyl-6-(propan-2-yl)-1,2-dihydropyridin-2-one
(1S,5R)-3-[(2-butyl-1H-imidazol-4-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(3-tert-butyl-1,2,4-oxadiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
4-(3,6-dimethylpyrazin-2-yl)phenol
(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-1-(oxolane-3-carbonyl)-decahydro-1,6-naphthyridine
5-methyl-N-[(4-methylphenyl)methyl]-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
methyl 6-cyclobutanecarbonyl-2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{1-[3-(2-ethoxyethoxy)benzoyl]piperidin-3-yl}benzoic acid
N-[2-(2-fluorophenoxy)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[4-(3-methylphenyl)phenyl]-1-(1,3-oxazole-5-carbonyl)piperidine-4-carboxamide
2-ethoxy-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)benzamide
5-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}pyrazin-2-ol
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
5-methoxy-3-[1-(pyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
N-[(3S,4R)-1-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
5-{[(2H-1,3-benzodioxol-5-ylmethyl)(methyl)amino]methyl}-N-(1,3-dimethyl-1H-pyrazol-5-yl)-1,3-thiazol-2-amine
4-(1-{1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]piperidin-4-yl}ethyl)morpholine
methyl 2-{[5-(4-fluorophenyl)-4-[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-yl]pyrimidin-2-yl]sulfanyl}acetate
(3aS,6aS)-5-[(2-chloro-5-fluorophenyl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-(pyridin-3-ylmethyl)piperidin-3-amine
4-phenyl-3-({1-[(2S)-piperidine-2-carbonyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenol
N-{7-methoxy-2-oxo-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1,2,3,4-tetrahydroquinolin-6-yl}methanesulfonamide