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{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
1-[(4-ethylphenyl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(1R,9aR)-1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-octahydro-1H-quinolizine
N4-[(2-amino-1,3-thiazol-4-yl)methyl]-N2,N2,5,6-tetramethylpyrimidine-2,4-diamine
methyl 3-[(3,4-dimethylphenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N'1-(2-hydroxyethyl)-N'1-[(2E)-3-phenylprop-2-en-1-yl]cyclopropane-1,1-dicarboxamide
1-(3-cyanopyridin-2-yl)-4-(2-phenoxyethyl)piperidine-4-carboxylic acid
N,1-diethyl-N-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
4-[4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carbonyl]-3-(propan-2-yl)piperazin-2-one
1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
3-{[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]methyl}phenol
5-(azocane-1-carbonyl)-2-[3-(1H-imidazol-1-yl)propyl]-2,3-dihydro-1H-isoindol-1-one
2-(morpholin-3-yl)-N-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)acetamide
1-({4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]phenyl}methyl)-1H-1,2,3,4-tetrazole
2-hydroxy-4-methyl-N-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
5-(oxolan-3-yl)-1-(2-phenoxyethyl)-4-phenyl-1H-imidazole
5-{4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carbonyl}-2-(pyridin-2-yl)pyrimidin-4-ol
3-{1-[(4-chloro-3-fluorophenyl)methyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
3-{[benzyl(methyl)amino]methyl}-1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
2-methyl-4-oxo-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
3,5-dimethoxy-N-({1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}methyl)benzamide
8-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N,N-diethylacetamide
1-[3-(dimethylcarbamoyl)pyridin-2-yl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(thiophene-3-carbonyl)piperidin-4-yl]propanamide
4-[1-(2-ethylbutyl)piperidin-4-yl]thiomorpholine
N-cyclopropyl-2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
7-(3-chlorophenyl)-4-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{4-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-{1-[1-(4-methanesulfonylphenyl)ethyl]-1H-imidazol-2-yl}benzoic acid
1-(4-fluorophenyl)-5-[(3,4,5-trimethoxyphenyl)methyl]-1H-1,2,4-triazole
6-(4-ethylpiperazin-1-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-(1,2,3-thiadiazole-4-carbonyl)piperidine
1-(oxolane-3-carbonyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
2-({2-[4-(cyclopropylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]phenyl}amino)acetic acid
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyrrolidine-3-carboxamide
3-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3H,4H-pyrido[4,3-d]pyrimidin-4-one
N'1-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
methyl[(1-methyl-1H-imidazol-5-yl)methyl][(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
N-(1-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperidin-4-yl)methanesulfonamide
5-methoxy-2-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridin-4-ol
N-[2-(ethylsulfanyl)phenyl]-4-[2-(morpholin-4-yl)ethyl]piperazine-1-carboxamide
2-({4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}methyl)quinolin-4-ol
4-(2-methoxyphenyl)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
N-[(3R,4S)-1-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-4-cyclopropylpyrrolidin-3-yl]methanesulfonamide
4-chloro-1-methyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
4-{[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]methyl}-1-propylpiperidine
1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-hydroxyethan-1-one