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1-{4-[2-(azocane-1-carbonyl)-4-chlorophenoxy]piperidin-1-yl}ethan-1-one
2-(dimethylamino)-2-(2-methylphenyl)-1-(1,4-oxazepan-4-yl)ethan-1-one
3-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-6-methylpyridazine
3-(3-methoxyphenyl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
4-{[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}-1-phenylpiperazin-2-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-hydroxypropanamide
4-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]-1λ6-thiomorpholine-1,1-dione
{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]methylamine
1-[6-hydroxy-4-(5-phenyl-1,2,4-oxadiazol-3-yl)-1,4-diazepan-1-yl]ethan-1-one
2-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetamido}-N-(2-fluoro-4-methylphenyl)propanamide
6-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-2-methyl-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
1-[1'-(1-ethylpyrrolidine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)-1,3-diazinane-2,4-dione
12-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
(1H-1,3-benzodiazol-2-ylmethyl)[(4-fluorophenyl)methyl](oxolan-2-ylmethyl)amine
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
3-(ethylsulfanyl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
2-{4-methyl-3-oxo-1H,2H,3H-pyrazolo[3,4-b]pyridine-6-carbonyl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one
2-(dimethylamino)-2-(2-fluorophenyl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)acetamide
3-[1-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1H-1,2,3-benzotriazole
3-[(3R,4S)-4-(morpholin-4-yl)-1-(phenylcarbamoyl)piperidin-3-yl]propanoic acid
5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
[3-(cyclopropylmethyl)-1-(3-methoxy-4-methylbenzoyl)piperidin-3-yl]methanol
1-[(3-chlorophenyl)methyl]-4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperazine
1-{1-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
8-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridin-3-ol
[(3-fluoropyridin-2-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
5-chloro-3-methyl-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
(4aR,8aS)-6-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-{[3-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
5-[(2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-3-(2-oxoazepan-1-yl)propanamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3,3,3-trifluoropropanamide
3-methyl-6-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyridazine
4-(methoxymethyl)-6-[4-(pyrazin-2-yl)piperazin-1-yl]pyrimidine
3-(5-methyl-1H-indol-3-yl)-4H-chromen-4-one
1-[3-(5-amino-3-methyl-1-phenyl-1H-pyrazol-4-yl)phenyl]ethan-1-one
5-(2,6-dimethoxyphenyl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1,2,4-triazin-3-amine
1-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
N-{[5-(methylsulfanyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
6-methyl-4-{4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
4-[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]-3-methylpiperazin-2-one
(1s,4s)-4-[4-(1,4-oxazepane-4-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexan-1-amine
1-[(2-methylpyrimidin-5-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
3-cyclopentaneamido-4-methyl-N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)benzamide
N-[(5-methoxy-1H-indol-2-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
1-(4-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}piperidin-1-yl)ethan-1-one
2-[4-(2-phenylethyl)-1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol