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N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-4-(trifluoromethyl)pyrimidin-2-amine
6-(4-ethylphenyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
7-(furan-3-ylmethyl)-N-[2-(1H-imidazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-cyclopropyl-1-[(4-ethylphenyl)methyl]-5-(1-methyl-1H-pyrazol-4-yl)-1H-1,2,4-triazole
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-(quinoxalin-6-ylmethyl)propanamide
5-acetyl-N-[(2-methoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)thiophene-3-carboxamide
5-(2-methoxyphenoxymethyl)-N-methyl-N-[1-(pyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
1-ethyl-4-{[(1R,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrrole-2-carbonitrile
N-[3-(2-fluorophenyl)propyl]oxane-2-carboxamide
2-[3-(4-cyclopentyl-1,4-diazepane-1-carbonyl)phenoxy]acetamide
methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
7-cyclopentyl-2-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)azepane-4-carboxamide
2-({1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}oxy)pyrimidine
N-{2-[3-(morpholin-4-ylmethyl)phenoxy]propyl}-1,3-thiazole-5-carboxamide
1,3-dimethyl-N-{2-[1-(2-methylpropyl)piperidin-2-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-cyclopentyl-N3-(3-methylbutyl)-4-oxo-N5-[2-(pyridin-4-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-ethyl-3-({1-[4-(1H-pyrazol-4-yl)butanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-amino-N-{2-[4-(furan-2-ylmethyl)morpholin-2-yl]ethyl}cyclopentane-1-carboxamide
2-(1H-imidazol-2-ylmethyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[4-(2,2-dimethylpropanamido)-3-methoxyphenyl]-3-sulfamoylthiophene-2-carboxamide
2-{6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}-1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazole
ethyl 2-(1-{2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamido}cyclohexyl)acetate
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[2-(pyridin-3-yl)ethyl]pyrrolidin-2-one
N-(2-methoxyethyl)-1-methyl-N-[(2-methylphenyl)methyl]azepane-2-carboxamide
4,6-dimethyl-2-{4-[3-(propoxymethyl)pyrrolidin-1-yl]piperidin-1-yl}pyrimidine
4-({4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}methyl)-2-(propan-2-yl)pyrimidine
4-chloro-2-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}phenol
4-{3,9-diazaspiro[5.6]dodecan-9-ylmethyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-{[3-(4-butyl-6-oxo-1,6-dihydropyrimidin-2-yl)phenyl]methyl}piperidine-3-carboxamide
1-ethyl-4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-4-phenylbutane-1,2-dione
N-cyclohexyl-4-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamido]piperidine-1-carboxamide
1-(4-{[2-(2-methyl-1H-indol-1-yl)ethyl]amino}piperidin-1-yl)ethan-1-one
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-1H-indazole-3-carboxamide
1-[3-(4-phenoxybenzoyl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(1-propylpiperidin-4-yl)piperidin-3-yl]piperazine
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-2-(1H-pyrazol-1-yl)-N-(pyridin-4-ylmethyl)benzamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
2-[5-(2-methyl-5-propylpyrimidin-4-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1-methyl-3-(propan-2-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1H-pyrazole-5-carboxamide
(1S,5R)-3-(2-methyl-4-phenylpyrimidine-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
1-{2-[(4-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(thiophen-3-ylmethyl)piperidine-4-carboxamide
(4aR,7aS)-1-(2-methylpropyl)-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2,5-dimethoxyphenyl)-3-[(3R)-3-hydroxypyrrolidin-1-yl]-3-oxopropanamide
3-[(2R,3R,6R)-5-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(pyridin-3-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
[1-(1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)piperidin-3-yl]methanol