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3-({[2-(1H-pyrazol-1-yl)phenyl]methyl}amino)-N-(pyridin-3-yl)propanamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}ethan-1-one
1-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
4-[7-(dimethyl-1,2-oxazole-4-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
1-(2,3-dimethylphenyl)-4-{[4-(2-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}piperazine
4-[7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,4-oxazepane
1-benzoyl-N-[(1-benzyl-1H-pyrazol-4-yl)methyl]piperidin-4-amine
7-cyclopentyl-2-(4-methylpiperazine-1-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[2-(3-fluorophenyl)ethyl]acetamide
6-fluoro-2-[(4-methanesulfonylpiperazin-1-yl)methyl]quinolin-4-ol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(5-methylthiophen-2-yl)methyl]piperidine-4-carboxamide
1-{4-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]thiophen-2-yl}ethan-1-one
N-cyclopropyl-4-methoxy-2-[(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)oxy]benzamide
N-tert-butyl-5-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
3-(1,3-benzoxazol-2-ylmethyl)-7-fluoro-3,4-dihydroquinazolin-4-one
(3S,4R)-1-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
2-cyclopropyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-methylpyrimidine
4-(3,3-diphenylpiperidine-1-carbonyl)-1λ6-thiane-1,1-dione
N-{[(3S,4S)-3-hydroxy-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl]methyl}morpholine-4-carboxamide
N4-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(morpholin-4-yl)ethyl]acetamide
7-(2-chloro-4-fluorophenyl)-1,2-dihydroisoquinolin-1-one
[(3S,4S)-4-(hydroxymethyl)-1-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}pyrrolidin-3-yl]methanol
2-methylpropyl 3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxylate
2-(3-hydroxyazetidine-1-carbonyl)-7-(prop-2-en-1-yl)-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide
1-(3-fluorophenyl)-4-(1H-imidazol-2-yl)-1H-pyrazole
1-[1-phenyl-3-(propan-2-yl)-1H-1,2,4-triazole-5-carbonyl]-2,3-dihydro-1H-indole
1-[2-(cyclohex-1-en-1-yl)ethyl]-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
ethyl 1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-4-(2-phenylethyl)piperidine-4-carboxylate
9-(1,4-dithiepan-6-yl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(furan-2-yl)phenyl]-1-(2-phenylethyl)piperidine-4-carboxamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
1-ethyl-5-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-1H-indole
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine
4-(1H-pyrazol-4-yl)-1-[4-(pyridin-4-yl)piperazin-1-yl]butan-1-one
4-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}piperazine-1-sulfonamide
1-{2-[ethyl(methyl)amino]acetyl}-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-(1H-1,3-benzodiazol-1-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
5-cyclopropanecarbonyl-1'-(3-ethyl-1,2-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
7-chloro-N-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-N-methyl-N-(piperidin-4-yl)butanamide
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]acetamide
2-{2-[(4-ethoxypyrimidin-2-yl)amino]ethyl}-6-methyl-3,4-dihydropyrimidin-4-one
1-ethyl-5-{methyl[(3-phenyl-1H-pyrazol-4-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(1R,5R)-3-[4-methoxy-3-(morpholin-4-yl)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane