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N-(butan-2-yl)-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-{[4-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]methyl}phenol
1-(2-methoxyphenyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
4-cyclopentyl-N-(5-acetamido-2-methoxyphenyl)-3-oxopiperazine-1-carboxamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[2-(pyridin-3-yloxy)propyl]acetamide
4,4,4-trifluoro-N-[(3R,4S)-1-(5-methyl-1,2,4-oxadiazol-3-yl)-4-(propan-2-yl)pyrrolidin-3-yl]butanamide
[(1,2-dimethyl-1H-imidazol-5-yl)methyl](methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(2R)-2-amino-4-methyl-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pentan-1-one
N-cyclopentyl-4-{4-[(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amino]piperidin-1-yl}benzamide
1-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{[5-(1-cyclohexylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}-4-methylpiperazine
N-methyl-1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(cyclohex-1-en-1-ylmethyl)-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(2H-1,3-benzodioxole-5-carbonyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-cyclopentanecarbonyl-N-methylpiperidine-4-carboxamide
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylacetamide
6-[(diethylamino)methyl]-N-[2-(1H-indol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{[(5-methylthiophen-2-yl)methyl]carbamoyl}pyrrolidine-2-carboxylate
2-(2,5-dioxoimidazolidin-1-yl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
N3-[2-(3-chlorophenyl)ethyl]-N5-[(2-fluorophenyl)methyl]-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-N-(propan-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
2-{1-[(2-aminopyridin-3-yl)methyl]pyrrolidin-3-yl}benzoic acid
1-{2-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-2-oxoethyl}-2-methyl-1,4-dihydroquinolin-4-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(1-propylpiperidin-4-yl)acetamide
1-ethyl-3-(hydroxymethyl)-N-(4-phenyl-1,2,3-thiadiazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
ethyl 4-(5-acetylthiophene-3-amido)piperidine-1-carboxylate
2-{1-[(2-chloro-6-fluorophenyl)methyl]pyrrolidin-3-yl}acetic acid
8-fluoro-N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}quinoline-2-carboxamide
2-methyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}thieno[3,2-d]pyrimidin-4-amine
3-{1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidin-4-yl}-1,3-oxazolidin-2-one
4-(4-ethyl-1H-pyrazol-5-yl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
4-(methoxymethyl)-6-[3-(1H-pyrazol-5-yl)phenyl]pyrimidine
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-methylpyrrolidine-2-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-methoxyacetamide
(3S,9aR)-3-[(benzyloxy)methyl]-8-(2-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}ethan-1-one
N-(furan-3-ylmethyl)-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
2-{[(2-hydroxy-6-methoxyquinolin-3-yl)methyl](methyl)amino}-N,N-dimethylpropanamide
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-2-(pyridin-4-yl)quinoline-4-carboxamide
(2S,4S)-N-ethyl-1-[(4-fluoro-2-methylphenyl)methyl]-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-cyclopropyl-5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]furan-2-carboxamide
4-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}-2,6-dimethoxyphenol
3-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-6-methylpyridazine
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(oxolan-2-ylmethyl)pyridin-2-amine
2-[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-2-methylpropane-1,3-diol
5-{4-[6-(piperidin-1-yl)pyrimidin-4-yl]piperazin-1-yl}-2,3-dihydropyridazin-3-one