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(3S,7S)-5-[2-(2-methoxyethoxy)acetyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
5-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrazine-2-carboxylic acid
5-(3-methylpyridine-4-carbonyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(3,5-difluorobenzoyl)-4-(2-methylpropyl)-1,4-diazepan-5-one
N-methyl-N-(2-phenyl-1-{1-[2-(1,3-thiazol-4-yl)acetyl]piperidin-4-yl}ethyl)thiophene-3-carboxamide
1'-[3-(2-methyl-1H-imidazol-1-yl)propyl]spiro[indene-1,4'-piperidine]
2-{[3-({1-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}carbamoyl)phenyl]amino}acetic acid
(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-6-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-decahydro-1,6-naphthyridin-2-one
methyl 4-{[(2-{1-[2-(methylsulfanyl)ethyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yl)ethyl]acetamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-(benzylamino)-1-(propan-2-yl)pyrrolidine-2-carboxamide
2,6-dihydroxy-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}benzamide
N-[4-(1,3-thiazol-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
2-{1-[1-(pyridin-3-yl)propan-2-yl]-1H-1,2,3-triazol-4-yl}-1H-1,3-benzodiazole
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-(4-fluorophenyl)-2-hydroxyethan-1-one
1-(pyridin-3-ylmethyl)-4-{[3-({1-[2-(trifluoromethyl)benzenesulfonyl]piperidin-4-yl}oxy)phenyl]methyl}piperazine
methyl (1R,3S,3aR,6aS)-5-benzyl-1-ethyl-4,6-dioxo-3-(1,3-thiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamide
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-(carbamoylmethyl)-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}piperidine-4-carboxamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(4-fluorophenyl)-1,4-diazepane
6-fluoro-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N,N-dimethyl-3-[(3S,4R)-1-(pyridin-2-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-[4-(trifluoromethyl)benzoyl]piperidine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2,5-dimethylfuran-3-carboxamide
4-{3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-3-ethylpiperazin-2-one
2-(cyclopropylmethyl)-8-[(4-methylthiophen-2-yl)sulfonyl]-2,8-diazaspiro[5.5]undecan-3-one
N3-cyclooctyl-N5-(cyclopropylmethyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(1H-1,2,4-triazol-5-ylmethyl)acetamide
N-(2-methoxyethyl)-7-(4-methoxypyrimidin-2-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[4-(4-phenyl-1H-imidazol-5-yl)phenyl]acetamide
2-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methylpyrazine
N-(furan-2-ylmethyl)-N'-[2-(methylsulfanyl)phenyl]-N-(prop-2-en-1-yl)butanediamide
6-({2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)-1,4-oxazepan-6-ol
N-(oxan-4-yl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
(2S,4S)-4-amino-N-methyl-1-[(3E)-4-phenylbut-3-enoyl]pyrrolidine-2-carboxamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine
3-({[3-(azepan-1-yl)propyl](methyl)carbamoyl}amino)-4-chloro-N-methylbenzamide
1-(4-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}thiophen-2-yl)ethan-1-one
N-benzyl-1-(2-hydroxyethyl)-5-(4,4,4-trifluorobutan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-3-(2-amino-1,3-thiazol-4-yl)propan-1-one
4-(cyclohexylmethyl)-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2-{[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}ethyl)acetamide
2-{1-[(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}pyridine
6-methoxy-3-(2-methoxyethyl)-3,4-dihydroquinazolin-4-one
1-(2-methoxybenzoyl)-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
2-[4-({3-ethyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)-2-methoxyphenoxy]acetamide
5-chloro-3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-[(3-methylquinoxalin-2-yl)methyl]pyrrolidin-3-amine