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1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-[1-(2-phenylethyl)pyrrolidin-2-yl]pyridine
8-[(2R)-2-amino-3-(4-chlorophenyl)propanoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-methyl-8-{2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4R)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
4-{[2-(cyclopropylmethyl)-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]methyl}-1H-imidazole
2-{octahydropyrrolo[1,2-a]piperazin-2-yl}-N,N-bis(prop-2-en-1-yl)acetamide
N-[2-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)propyl]-2H-1,3-benzodioxole-5-carboxamide
[2-(1H-indol-1-yl)ethyl](methyl){[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
(2S)-2-amino-1-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pentan-1-one
2-{4-[(2-aminopyrimidin-5-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
5-(2-methoxy-2-phenylacetyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(methylsulfanyl)-4-{3-[1-(1,3-thiazol-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
N-{7-oxo-5-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}thiophene-2-carboxamide
2-methyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-4-carboxamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]methanesulfonamide
2-(4-{[3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenoxy)acetic acid
N-(2,3-dihydroxypropyl)-N-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
(3aR,6aR)-2-[2-(4-fluorophenyl)acetyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]pyrrolidin-3-yl}piperidine
1-{2-[2-(2,5,7-trimethyl-1H-indol-3-yl)acetamido]ethyl}piperidine-3-carboxamide
1-ethyl-4-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}pyrrolidin-2-one
N-[3-(2-methoxyphenyl)propyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-(dimethylamino)-N-methyl-2-(2-methylphenyl)-N-(1H-pyrazol-3-ylmethyl)acetamide
butyl (1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxylate
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-phenyl-4-{[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl}-1H-1,2,3-triazole
2-[2-(2-fluorophenyl)ethyl]-4-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
2-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]benzene-1,3-diol
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
methyl 4-(5-{[2-(2-hydroxyethyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
2-[3-(3-methoxypropyl)piperidine-1-carbonyl]thiophen-3-amine
2-[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-5-carboxylic acid
9-(2,3-dihydro-1H-indene-1-carbonyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(4-chloro-3-fluorophenyl)-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]acetic acid
9-(3,4-dimethylbenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3,5-difluoropyridin-2-amine
4-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-3-yl)benzoic acid
4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyrimidine
1-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}isoquinoline
2-(2-acetyl-4,5-dimethoxyphenyl)-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-({5-[1-(2-aminoethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
1-[3-(1H-1,3-benzodiazol-2-yl)azetidin-1-yl]-2-hydroxy-4-(methylsulfanyl)butan-1-one
3-(aminomethyl)-4-(2,3-dichlorophenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
2-(5-fluoro-2-methylphenyl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
(3aR,7aS)-5-methyl-2-(2-propylpyridine-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole