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2-(4-{[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]methyl}-2-chlorophenoxy)acetamide
3-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-[3-(morpholin-4-yl)propyl]urea
3-(2-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
(1S,5R)-N-(3-cyanophenyl)-3-[(dimethylcarbamoyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-{[3-(difluoromethoxy)phenyl]methyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(4-phenylpiperazin-1-yl)-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]propan-1-one
7-(cyclobutylmethyl)-2-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
(2R,6R)-4-[(4-fluoro-2-methylphenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-{2-[(4-methylphenyl)sulfanyl]ethyl}pyrimidin-2-amine
3-(1,2-oxazinan-2-yl)-1-(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidin-1-yl)propan-1-one
1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
5-{2-[(pyridin-3-ylmethyl)amino]ethyl}-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-methyl-N-(propan-2-yl)acetamide
methyl 6-(1H-indol-4-yl)pyridine-3-carboxylate
(1-{3-[1-(difluoromethyl)-5-methyl-1H-pyrazol-4-yl]phenyl}ethyl)dimethylamine
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-(pyridine-3-carbonyl)piperidin-4-amine
N-methyl-2-(N-methyl-1-{2-[(quinolin-6-yloxy)methyl]-1,3-oxazol-4-yl}formamido)acetamide
N-(propan-2-yl)-1-[(1s,4s)-4-{[(2,4-dimethoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-ethyl-2-methylpyrimidine
5-(2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-ethyl-2-(8-methoxy-2-methylquinolin-5-yl)pyrimidin-4-amine
3-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-methyl-1-(2-methyl-1-benzofuran-7-yl)urea
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
3-methyl-1-{3-[(phenylsulfanyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}but-2-en-1-one
8-cyclopropanecarbonyl-2-(4-methoxybenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
[(3R,4R)-1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
4-ethyl-3-{1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
{4-[(dimethylamino)methyl]-1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}methanol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-[(prop-2-en-1-yl)amino]benzamide
2-{4-[1-(4-methyl-1,3-oxazole-5-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
ethyl 1-{[3-(benzyloxy)phenyl]methyl}-4-(2-methoxyethyl)piperidine-4-carboxylate
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-2-oxo-1,2-dihydroquinazoline-4-carboxamide
(3R,5S)-N3-(4-fluorophenyl)-1-(2-methylpropyl)-N5-[2-(morpholin-4-yl)ethyl]piperidine-3,5-dicarboxamide
4-hydroxy-N-(2-methoxyethyl)-2-(4-methylphenyl)-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide
2-{4-[7-methyl-3-(morpholin-4-ylmethyl)quinolin-2-yl]piperazin-1-yl}ethan-1-ol
1-[2-(dimethylamino)ethyl]-N-[(6-methylquinolin-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N3-cyclooctyl-N5-[(3-methylphenyl)methyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
6-[(2-hydroxyethyl)amino]-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide
4-{[(2-{4-[5-(methoxymethyl)thiophene-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]carbamoyl}pyridin-1-ium-1-olate
N-[(2R,4R,6S)-2-(3-hydroxyphenyl)-6-(2,4,5-trimethylphenyl)oxan-4-yl]acetamide
4-(2-methyloxane-2-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
5-{4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2-ethylpyrimidine
6-(methylamino)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1-[(2-methoxyphenyl)methyl]piperidin-2-one
5-(oxolane-3-carbonyl)-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(1S,6R)-9-(2-hydroxy-4-methoxybenzoyl)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one