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(isoquinolin-5-ylmethyl)({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
2-amino-4-(2-aminopyrimidin-5-yl)-6-[3-(trifluoromethyl)phenyl]pyridine-3-carbonitrile
(2-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl][(5-methylthiophen-2-yl)methyl]amino}ethyl)dimethylamine
N-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-{[1-(dimethylamino)cycloheptyl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
1-[3-(3-methoxyphenoxy)azetidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
8-[(4-fluoro-3-methoxyphenyl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S)-2-(hydroxymethyl)-N-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-1-carboxamide
N-{4-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-4-oxobutyl}acetamide
N-[2-(oxolan-2-ylmethoxy)phenyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(3-chlorophenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]thiophene-3-carboxamide
N-cyclopropyl-4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperazine-2-carboxamide
1-[2-({methyl[2-(morpholin-4-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
(2S)-2-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]-3-phenylpropanamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-chlorophenyl)-1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(1S,5R)-3-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]isoquinoline
4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-[(2-methylphenyl)methyl]-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazine
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-5H-thiochromeno[4,3-b]pyridine-3-carbonitrile
N-{2-[2-(1,1-dioxo-1λ6-thiolan-3-yl)ethyl]phenyl}-2-methoxyacetamide
3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole
3-ethyl-3-(hydroxymethyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
N-(4-methylphenyl)-3-oxo-3-[4-(pyridin-2-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propanamide
3-[3-(3-phenylpropanoyl)piperidine-1-carbonyl]benzonitrile
N-methyl-5-(phenoxymethyl)-N-[1-(pyridin-3-yl)propyl]-1H-pyrazole-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(3-methoxyphenyl)-1,3-benzoxazole-6-carboxamide
ethyl 1-(5-chloro-2-methoxybenzenesulfonyl)-4-(cyclopropylmethyl)piperidine-4-carboxylate
(4aR,7aS)-1-[2-(4,4-difluoropiperidin-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(1-benzylpiperidin-4-yl)-N-[2-(pyridin-3-yl)ethyl]piperidine-3-carboxamide
2-(5-{[3-(pyridin-4-yl)azetidin-1-yl]methyl}-1,2-oxazol-3-yl)pyridine
(2S)-2-{4-[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]-1H-1,2,3-triazol-1-yl}butanoic acid
7-[(2,3-dimethoxyphenyl)methyl]-2-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-[(4-cyclohexyl-1,4-diazepan-1-yl)methyl]-8-fluoroquinolin-4-ol
N-(butan-2-yl)-N-[(2-fluorophenyl)methyl]-2-methyl-5-sulfamoylbenzamide
4-[4-(cyclohexylmethyl)-3-oxo-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl]-1,4-diazepane-1-carbaldehyde
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
3-hydroxy-3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
1-(2-{[4-(methoxymethyl)phenyl]formamido}ethyl)piperidine-3-carboxamide
1-[(4-fluorophenyl)methyl]-4-(1-methylazepane-2-carbonyl)-1,4-diazepane
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
methyl (1S,3S,3aR,6aS)-5-methyl-4,6-dioxo-1-phenyl-3-(pyridin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
3-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-[(1R)-1-(4-fluorophenyl)ethyl]urea
3,3-diphenyl-1-(1H-pyrrole-3-carbonyl)piperidine
5-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]thiophene-2-carboxamide
2-ethyl-4-{[4-(oxan-4-yl)piperazin-1-yl]methyl}pyrimidine
5-(propan-2-yl)-N-[2-(pyridin-2-yl)ethyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide