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1-{1-[1-(4-chlorophenyl)cyclopropanecarbonyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
3-(3-fluorophenyl)-4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-6-oxo-1,6-dihydropyridazine-3-carboxamide
5-[4-(1H-pyrazol-5-yl)phenyl]pyrazin-2-amine
1-(5-{2-[2-(ethylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}-1-methyl-1H-1,3-benzodiazol-2-yl)ethan-1-ol
N-[(3-chlorophenyl)methyl]-3-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl}propanamide
7-(1,3-benzothiazol-2-yl)-4-(pyrimidin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-imidazole
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-3-(3-hydroxy-3-methylbutyl)benzamide
8-(1,3-benzothiazol-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-chloro-2-methoxy-5-methylphenyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
5-[(1-butyl-1H-1,2,4-triazol-5-yl)methyl]-2-methyl-1H-1,3-benzodiazole
1-(1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-2-yl)pyrrolidine
1-[1-(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)ethyl]-4-methylpiperazine
7-(3-chlorophenyl)-4-(oxolan-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-methoxy-2-{3-methyl-3,9-diazaspiro[5.6]dodecane-9-carbonyl}phenol
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-2-(4-propanoylphenoxy)acetamide
2-amino-1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
1-(6-methoxypyridin-3-yl)isoquinoline
3-(5-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
(1S,5R)-3-(pyrazine-2-carbonyl)-6-(pyrrolidine-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-({[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}methyl)benzene-1-sulfonamide
6-fluoro-2-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(2-methoxyphenyl)-2-methylpiperazine
3-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-yl]-N-[(2,4-dimethoxyphenyl)methyl]propanamide
10-methoxy-5-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-ethyl-5-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}pyrimidin-2-amine
2-({[(1-benzyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)pyridine-3-carboxylic acid
3-(2-methoxyphenoxy)-1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)azetidine
N-(4-fluorophenyl)-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-amine
2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-5-(propan-2-yl)pyrimidine
2-amino-N-[2-(1,3-thiazol-4-yl)ethyl]-4-(trifluoromethyl)pyrimidine-5-carboxamide
5-cyclohexaneamido-N-[(2,3-difluorophenyl)methyl]-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
1-(4-cyclopentylpyrimidin-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(2S,4S)-4-amino-N-ethyl-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidine-2-carboxamide
3,6-dimethyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
(3S,4R)-3-cyclopropyl-N,N-dimethyl-4-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-amido}pyrrolidine-1-carboxamide
[(3R,4S)-1-[(3,5-dimethoxyphenyl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N,N-dimethyl-4-({2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)oxan-4-amine
N-[(2-fluorophenyl)methyl]-2-{[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]amino}acetamide
6-(pyrrolidin-1-ylmethyl)-4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-1,4-oxazepan-6-ol
9-(3-ethoxybenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(benzylsulfamoyl)(methyl){[2-(trifluoromethyl)phenyl]methyl}amine
(1-{[1-(6-fluoro-1H-1,3-benzodiazole-2-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanamine
(3S,4R)-4-(4-fluorophenyl)-1-[5-(methoxymethyl)thiophene-2-carbonyl]pyrrolidine-3-carboxylic acid
(2E)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-phenyl-N-(propan-2-yl)prop-2-enamide
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-methyl-3-(pyrrolidin-1-yl)propan-1-one
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
(3aS,6aS)-5-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide