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2-{2-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
4-[1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]butanoic acid
4-methyl-2-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
N-benzyl-1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
4-(isoquinoline-5-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-ethyl-N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)pyrimidine-5-carboxamide
1-[4-(difluoromethoxy)-2-methylphenyl]-3-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]urea
ethyl 1-(oxan-2-ylmethyl)-1H-imidazole-2-carboxylate
4-{2-[4-(4-ethyl-5-methylpyrimidin-2-yl)piperazin-1-yl]ethyl}morpholine
(4aS,8aR)-6-(4-fluoro-3-methylbenzoyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
(4aS,8aR)-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
3-cyclohexyl-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
2-cyclohexyl-6-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-1,3-benzoxazole
4-{2-[(6-phenylpyridazin-3-yl)oxy]hex-5-en-1-yl}-1,4-oxazepane
2-methyl-1-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}piperazine
3-(1H-1,2,3-benzotriazol-1-yl)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]propan-1-one
N-(2,3-dihydroxypropyl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-(2-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}quinolin-5-yl)acetamide
3-[1-(1,3-thiazol-2-yl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
4-[1-({2-[(carboxymethyl)(methyl)amino]pyrimidin-5-yl}methyl)piperidin-3-yl]benzoic acid
1-ethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-oxopyrrolidine-3-carboxamide
N-[1-(2-chlorophenyl)ethyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
[(3R,5R)-1-(2-methyl-1,3-benzothiazole-6-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-1-(morpholin-4-yl)propan-1-one
N-butyl-1-{1,3-dioxo-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-3-carboxamide
N-(furan-2-ylmethyl)-1,3-dimethyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-1H-pyrazole-5-carboxamide
N-[3-(azepan-1-yl)-2-hydroxypropyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2,3-dimethyl-1H-indole
3-amino-N-{2-[4-(furan-2-ylmethyl)morpholin-2-yl]ethyl}-1H-1,2,4-triazole-5-carboxamide
N-[(1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-3-yl)methyl]methanesulfonamide
N-tert-butyl-2-methyl-3-[2-(1H-pyrazol-1-yl)butanamido]benzamide
1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-(methylsulfanyl)ethan-1-one
4-[4-(1-benzothiophene-5-carbonyl)piperazin-1-yl]-6-methylpyrimidin-2-amine
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-ol
N-{[1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidin-4-yl]methyl}acetamide
N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
1-(2,5-dimethylpyrimidin-4-yl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
(3R,9aR)-8-[(3-methoxyphenyl)methyl]-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-amino-1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,N-diethyl-2-oxoacetamide
2-(2-methoxyphenyl)-1-[2-(morpholine-4-carbonyl)piperazin-1-yl]ethan-1-one
2-ethyl-8-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
3-({[4-(ethylamino)pyrimidin-2-yl]amino}methyl)-1λ6-thiolane-1,1-dione
3-(2,4-dimethoxybenzoyl)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidine
3-[(4-methoxyphenyl)methyl]-1-methyl-8-{[4-(2-methylphenyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
4-[(5-oxopyrrolidin-2-yl)methyl]-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
2-(4-ethylpiperazin-1-yl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[3-(5-methylfuran-2-yl)butyl]piperidine
2-[8-(oxane-4-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid