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4-methyl-N-{[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl}pyrimidin-2-amine
2-methyl-2-[2-(3-methylpiperidin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]propanoic acid
2-[3-(5-methylfuran-2-yl)-5-(pyridin-2-yl)-1H-1,2,4-triazol-1-yl]acetic acid
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
2-ethyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2H-1,2,3,4-tetrazol-5-amine
2-(4-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-ol
4-benzoyl-3-benzylpiperazin-2-one
2-(2-{[3-(dimethyl-1,3-thiazol-2-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
6-(4-fluorophenyl)-2-[2-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
4-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
1,4-dimethyl 2-({1-[4-(4-methoxybenzamido)phenyl]piperidin-4-yl}amino)butanedioate
4-(furan-3-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(4-fluorophenyl)-N-[phenyl(pyridin-2-yl)methyl]-1H-pyrazole-5-carboxamide
(1S,5R)-3-benzoyl-6-(benzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonane
2-methoxy-4-(5-methoxy-1H-indol-2-yl)pyridine-3-carbonitrile
5-({[(6-hydroxy-1,4-oxazepan-6-yl)methyl]amino}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-({1-[(6-chloro-2H-chromen-3-yl)methyl]piperidin-3-yl}methyl)furan-2-carboxamide
2-hydroxy-4-(methylsulfanyl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}butanamide
2-[(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]pyridine-4-carbonitrile
1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-N-cyclopropylpiperazine-2-carboxamide
2-(4-fluorophenyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
methyl 3-[({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)carbamoyl]propanoate
3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-N,N-dimethylaniline
1-[3-(methylsulfanyl)phenyl]-3-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
4-[(3,5-dichloropyridin-4-yl)methyl]-1-(2-methoxyphenyl)piperazin-2-one
1-[(2,6-difluorophenyl)methyl]-4-[(dimethylamino)methyl]azepan-4-ol
3-{[1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)pyrrolidin-3-yl]methyl}benzoic acid
(1R,5R)-6-(cyclobutylmethyl)-3-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-(2-chlorophenyl)-2-methyl-N-[(5-methylpyrazin-2-yl)methyl]furan-3-carboxamide
4-(2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-1H-pyrrol-1-yl)benzonitrile
2,6-dimethyl-8-[(1-phenylcyclopropyl)amino]octan-2-ol
2-(3,4-dimethoxyphenyl)quinoxaline
N3-[2-(3-fluorophenyl)ethyl]-N5-[(3-methylphenyl)methyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
4,4,4-trifluoro-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
2-[3-oxo-9-(5-propyl-1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
3-benzoyl-1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine
4-({2-[1-(3-methoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(1-hydroxybutan-2-yl)-2-{imidazo[1,2-a]pyridin-3-yl}-N-[(5-methylthiophen-2-yl)methyl]acetamide
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
1-[4-(2-methanesulfonylethyl)piperazin-1-yl]-3-(2-methyl-1H-indol-1-yl)propan-1-one
N-(4-{2-methyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}phenyl)ethane-1-sulfonamide
N-[(3R,5S)-1-cyclopropanecarbonyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-5-propyl-1,2-oxazole-4-carboxamide
N-{[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]methyl}-2-(methylsulfanyl)pyridine-3-carboxamide
1-[3-(hydroxymethyl)-3-(2-methylpropyl)piperidin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
2-(2-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-N,1-dimethyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-cyclooctylpiperidin-3-ol
2,2-dimethyl-3-[methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})amino]propan-1-ol