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8-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-[4-(3-fluorophenyl)benzoyl]-4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
4-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,7aR)-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1-[4-(pyridin-3-yl)pyrimidin-2-yl]pyrrolidin-3-yl}acetamide
4-[(6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-yl)methyl]morpholine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
4-[2-(2-chlorophenoxy)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-hydroxy-N-[1-(pyrazin-2-yl)propan-2-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-(adamantan-2-yl)-N'-(4-methylphenyl)propanediamide
4-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepane-1-carbaldehyde
2-[(3S,4R)-3-cyclopropyl-4-[3-(trifluoromethyl)-1H-pyrazole-5-amido]pyrrolidin-1-yl]acetic acid
6-oxo-N-(prop-2-en-1-yl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane-2-carboxamide
N-[2-(2-methyl-1-phenyl-1H-indol-3-yl)ethyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[(2R)-1,1,1-trifluoro-3-methylbutan-2-yl]propanamide
N-(2-methoxyethyl)-3-(1,2-oxazinan-2-yl)-N-(3-phenylprop-2-yn-1-yl)propanamide
4-{[(3-hydroxypiperidin-3-yl)methyl]sulfamoyl}-N-propylbenzamide
[1-(5-chloropyridin-2-yl)-3-ethylpiperidin-3-yl]methanol
2-(4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
3-[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]-1,2-dihydropyrazin-2-one
N-(1-{1-[(2,6-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
8-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
9-(3-chloro-4-fluorobenzoyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
(5S,9aS,9bS)-5-[5-(methoxymethyl)furan-2-yl]-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-ethyl-4-methyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1,3-thiazole-5-carboxamide
4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-2,5-dimethyl-1,3-oxazole
1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
N,N-dimethyl-5-({4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)-1,3-thiazol-2-amine
1-[6-(aminomethyl)-2-methylpyrimidin-4-yl]-N,N-diethylpiperidine-3-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]quinoxaline-6-carboxamide
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
N-{2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}methanesulfonamide
3-chloro-6-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-benzyl-8-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
4-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-2-(4-fluorophenyl)morpholine
6-{3-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
N-ethyl-5-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}pyrimidin-2-amine
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-4-(piperidin-1-yl)butanamide
1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-[(3-fluorophenyl)methyl]piperazine
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-({2-[2-(cyclopropylcarbamoyl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)benzoic acid
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrrolidin-3-yl]methanol
3-[({[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}amino)methyl]-N,N-dimethylpyridin-2-amine
ethyl 4-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}piperidine-1-carboxylate
[(3R,4R)-1-(2-methyl-1,3-thiazole-4-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-methyl-5-({methyl[(5-propyl-1H-pyrazol-3-yl)methyl]amino}methyl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-(methoxymethyl)-1-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidine
2-(2-aminoethyl)-N-(cyclopropylmethyl)quinazolin-4-amine