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2-(4-{1-[(3S,4R)-4-methoxyoxolan-3-yl]-4-phenyl-1H-imidazol-5-yl}phenoxy)ethan-1-ol
2-methyl-4-(3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)butan-2-ol
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
(1R,3S,5S)-8-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane
N3-(3-{[(2-chlorophenyl)methyl]sulfanyl}propyl)piperidine-1,3-dicarboxamide
3-amino-1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)pyrrolidine-3-carboxylic acid
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}thiophene-2-carboxamide
N-methyl-2-(2-propyl-1H-1,3-benzodiazol-1-yl)-N-[2-(pyridin-2-yl)ethyl]propanamide
1-{pyrazolo[1,5-a]pyridine-7-carbonyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
7-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
benzyl({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)methylamine
1-{2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethyl}pyrrolidin-2-one
2,6-dimethoxy-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrimidine-4-carboxamide
6,6-dimethyl-1-phenyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-chloro-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-amine
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-N-propyl-1,3-oxazole-4-carboxamide
2-{[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
N-[(2-chloro-4-fluorophenyl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
3-(1H-1,2,3-benzotriazol-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}azepan-4-amine
methyl 3-(2-chlorobenzenesulfonamido)-5-{[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetamido]methyl}benzoate
1-(2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
N,1-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1H-indazole-3-carboxamide
N-[2-(4-chlorophenyl)ethyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
N-{1-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
2-[2-({3-azaspiro[5.5]undecan-9-yl}amino)ethyl]-3,4-dihydroquinazolin-4-one
1-methyl-1'-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
1-[1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-2-phenylethan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylquinoline-2-carboxamide
4-benzyl-3-[1-(1,2-oxazole-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(2-chlorophenyl)methyl]-N-methyl-N-[1-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
7-chloro-2-(2-methoxyphenyl)-3-[(4-methylpiperazin-1-yl)methyl]quinoline
2-chloro-6-methyl-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}benzamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-azaspiro[5.5]undecan-9-amine
(1H-1,3-benzodiazol-2-ylmethyl)bis(1,3-oxazol-4-ylmethyl)amine
2-{2-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-4-methylphenoxy}acetamide
[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)(quinolin-2-ylmethyl)amine
N,4-dimethyl-2-{9-methyl-3,9-diazaspiro[5.6]dodecane-3-carbonyl}aniline
(3aS,7aR)-2-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
5-(2-chloro-4-fluorophenoxymethyl)-N-(oxolan-2-ylmethyl)-N-propyl-1,2-oxazole-3-carboxamide
2-(2H-1,3-benzodioxol-4-yl)-1-[(2,6-difluorophenyl)methyl]-1H-imidazole
5-(3-{[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propyl)-1,3,4-thiadiazol-2-amine
2-(methylamino)-1-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
4-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-4-oxo-N-phenylbutanamide
(3S,7S)-5-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-(4-{[(4-cyclohexylphenyl)carbamoyl]amino}piperidin-1-yl)acetamide
3-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrazol-5-amine