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methyl 6-(4-hydroxyphenyl)pyridine-3-carboxylate
1-(azepan-1-yl)-3-[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]propan-1-one
1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-[(4-amino-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidin-2-yl)sulfanyl]-N,N-dimethylacetamide
5-(1H-indol-1-ylmethyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1H-pyrazole-3-carboxamide
3-[(3S,7S,8aS)-3-(1H-indol-3-ylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,3-dichlorophenyl)urea
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-[2-(pyridin-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{2-[5-(pentan-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
N-cyclopentyl-1-ethyl-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-3-carboxamide
1-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperidin-3-ol
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
2-(3-hydroxypropyl)-9-(3-methoxy-4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N,1-dimethyl-6-oxo-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1,6-dihydropyridine-3-carboxamide
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-(2-chlorophenyl)-1-(4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-hydroxyethan-1-one
ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)[3-(methylsulfanyl)propyl]amine
7-(furan-3-carbonyl)-N-(1H-imidazol-2-ylmethyl)-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
8-(6-methoxypyrimidin-4-yl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-{4-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]morpholin-3-yl}acetic acid
ethyl(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-3-(1-methylpiperidin-3-yl)propanamide
2-acetyl-8-methanesulfonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-benzofuran-5-carboxamide
1-benzyl-5-(cyclooctylamino)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-{[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl](phenyl)methyl}-1,3,4-thiadiazol-2-amine
2-{1-cyclopentyl-4-[(3,7-dimethyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
ethyl 4-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]piperidine-1-carboxylate
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
8-fluoro-4-oxo-N-(2,2,2-trifluoroethyl)-1,4-dihydroquinoline-3-carboxamide
(1,3-benzothiazol-2-ylmethyl)({[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
4-(1-methylpyrrolidine-3-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)pyridin-2-amine
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
2-[(3R,4S)-3-(2-carboxyethyl)-4-(morpholin-4-yl)piperidin-1-yl]-6-methylpyrimidine-4-carboxylic acid
3-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
2-[1-(2-methyl-1,3-benzothiazol-6-yl)-5-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-3-yl]acetamide
methyl 3-[(2,6-difluorophenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-({[1-(cyclohex-1-en-1-yl)ethyl]amino}methyl)-4-hydroxyquinoline-6-carboxamide
2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(propan-2-yl)acetamide
3-(2-ethyl-1H-1,3-benzodiazol-1-yl)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyphenoxy)piperidine
N-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazine-1-carboxamide
3-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
(1R,5S,8R)-8-methoxy-3-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3-azabicyclo[3.2.1]octane
2-(2,3-dihydro-1H-inden-1-yl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}acetamide
1-(2-{5-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)pyrrolidin-2-one
2-(morpholin-4-ylmethyl)-N-[3-(prop-2-en-1-yloxy)phenyl]-1,4-oxazepane-4-carboxamide
(1-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)methanol