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(1R,5S,6R)-3-[(2,2-dimethyloxan-4-yl)methyl]-N-[(5-methylpyrazin-2-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
5-[1-(2-cyclohexylacetyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
5-phenyl-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-2-one
2-amino-7-[2-(pyrrolidin-1-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-methyl-3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-4,5,6,7-tetrahydro-1H-indazole
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(3-methylbut-2-en-1-yl)piperidine
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
(3S,5R)-5-(cyclopropylcarbamoyl)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidine-3-carboxylic acid
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)ethan-1-one
5-{3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2-(propan-2-yl)pyrimidine
1-phenyl-N-({1-[2-(thiophen-2-yl)acetyl]piperidin-3-yl}methyl)methanesulfonamide
2,6-dimethyl-N-[1-(1,3-thiazol-5-yl)propan-2-yl]quinoline-4-carboxamide
2-[(1-ethylpyrrolidin-2-yl)methyl]-3-oxo-N-(pyrimidin-4-ylmethyl)-2,3-dihydro-1H-isoindole-5-carboxamide
ethyl 4-[2-(2-aminoethyl)morpholine-4-carbonyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
4-(5-{1-ethyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}-1H-pyrazol-3-yl)phenol
N-cyclopropyl-N-{[6-(2,5-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-4-(trifluoromethyl)benzamide
3-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
2-(3-methoxypropyl)-9-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-5-(propan-2-yl)-1,2-oxazole
3-(1H-pyrazol-1-yl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-(1-methyl-1H-imidazole-2-carbonyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine
8-[(4-methoxyphenyl)methyl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
1-{7,7-dimethyl-5-[(6-methylpyrimidin-4-yl)amino]-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-ol
3-[(dimethylamino)methyl]-N-(3-fluoro-4-methylphenyl)-3-(hydroxymethyl)piperidine-1-carboxamide
2-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-5-methoxy-4H-pyran-4-one
[1-(2-methylpyrimidin-4-yl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
2-(2,3-dihydro-1H-inden-1-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-(2-fluoro-4-methoxyphenyl)-4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carboxamide
3-methyl-8-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanoyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5R)-3-(2,4-difluorobenzenesulfonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1H-1,2,3-triazole-5-carboxamide
4-(2-ethoxypyridin-3-yl)-6-ethyl-N,N-dimethylpyrimidin-2-amine
1-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-1,4-diazepane-6-carboxylic acid
1-(3-methoxyphenyl)-6-methyl-4-[2-(pyridin-3-yl)acetyl]piperazin-2-one
ethyl 5-({[1-(furan-2-yl)ethyl]amino}methyl)-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
N-[(3S,4R)-1-(1-benzofuran-2-ylmethyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
3-[1-(3-aminothiophene-2-carbonyl)piperidin-3-yl]-N,N-dimethylpropanamide
3-[(2R,5S)-2,5-dimethylpyrrolidine-1-carbonyl]-5-(2-methoxyphenoxymethyl)-1H-pyrazole
{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}(benzylsulfamoyl)amine
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-(1H-pyrazol-1-yl)butan-1-one
2-[(2,3-dichloro-6-fluorophenyl)methyl]-5-(dimethylamino)-2,3-dihydropyridazin-3-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)cyclopentanecarboxamide
3-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
8-methoxy-2-{[1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxy}quinoline
2-[5-(3-methyl-3-phenylpiperidine-1-carbonyl)-1H-1,3-benzodiazol-1-yl]ethan-1-ol
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxamide