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3-(3,4-dimethyl-1H-pyrazol-5-yl)-N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}propanamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(morpholin-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
2-{[1-(pyrazin-2-yl)propan-2-yl]amino}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-2-oxoacetamide
{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}bis(prop-2-en-1-yl)amine
3-[4-(4-fluorophenyl)piperazin-1-yl]-5-(2-methylphenyl)-1,2,4-triazine
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-5-(naphthalen-1-yl)-1,2,4-triazin-3-amine
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-3-[(2-methylpyrrolidin-1-yl)sulfonyl]benzamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1-propyl-1H-pyrazole-5-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[5-methyl-2-(methylamino)phenyl]formamido}acetic acid
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
4-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-ethyl-3-methyl-1H-pyrazole
N-[(2,4-dihydroxyphenyl)methyl]-2-(dimethylamino)-2-(3-methylphenyl)acetamide
6-methyl-4-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-(4-methylpiperazin-1-yl)-6-{1H-pyrrolo[2,3-b]pyridin-4-yl}quinazoline
6-methyl-2-oxo-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1,2-dihydropyridine-4-carboxamide
6-[4-(acetamidomethyl)piperidin-1-yl]pyridine-2-carboxylic acid
N-(9H-fluoren-9-yl)-6-({methyl[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
[(3R,4R)-1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
4-(5-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl)morpholine
1-(carbamoylmethyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]piperidine-3-carboxamide
3-[(1-benzylpiperidin-4-yl)oxy]-N-cyclopropyl-4-methoxybenzamide
N-[(3R,5S)-1-(cyclopentylmethyl)-5-(diethylcarbamoyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
(2S)-2-amino-4-[1-(carboxymethyl)-3-[(3-chlorophenyl)methyl]-1H-1,2,4-triazol-5-yl]butanoic acid
1-[(2-methoxyphenyl)methyl]-6-oxo-N-[3-(pyridin-3-yl)propyl]piperidine-3-carboxamide
methyl 4-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
2-[4-carbamoyl-4-(piperidin-1-yl)piperidin-1-yl]-2-(2,4-dimethylphenyl)acetic acid
(1R,7S)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(2-ethylbutyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-4-methylbenzamide
2-[benzyl(methyl)amino]-N-(1,3-dihydroxypropan-2-yl)-2,3-dihydro-1H-indene-2-carboxamide
3-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholine-4-carbonyl)pyridin-2-ol
1-methyl-N-{[4-(piperidine-1-carbonyl)phenyl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-{[(3-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}-4-methoxyphenyl)methyl]amino}-2,2-dimethylpropan-1-ol
propan-2-yl 2-chloro-5-(2-acetamidoacetamido)benzoate
2-{[7-(2,1,3-benzoxadiazol-4-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
2-[3-(2-ethoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-6-methylpyridine-3-carbonitrile
1-cyclohexyl-5-(2,6-difluorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
2-[2-(2,4-dimethylphenoxy)ethyl]-6-fluorobenzamide
2-(2-hydroxyethyl)-8-[2-(methylamino)pyridine-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-cyclobutanecarbonyl-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
3-(azepane-1-carbonyl)-N-methyl-N-(oxan-4-yl)benzene-1-sulfonamide
(1R,2R)-2-[({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-methylcyclohexan-1-ol
3-[2-(2-phenylethyl)morpholine-4-carbonyl]pyridin-1-ium-1-olate
N-(2-{[5-(2-methylphenyl)-4-(4-methylphenyl)pyrimidin-2-yl]amino}ethyl)acetamide
6-[4-(trifluoromethoxy)phenyl]-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
2-amino-6-(2,2-dimethyloxan-4-yl)-5-methyl-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
3-(cyclopropylmethyl)-1-(3-fluoro-5-methylphenyl)-3-(2-methoxyethyl)urea
2-(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)-4-methoxypyrimidine