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[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl][(3-ethyl-1,2-oxazol-5-yl)methyl]methylamine
(5S,9aS,9bS)-5-(1-methyl-1H-pyrazol-4-yl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-(2,5-dioxoimidazolidin-4-yl)-N-{[2-(3-methylphenyl)-1,3-thiazol-4-yl]methyl}propanamide
N,N-dimethyl-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonamide
7-cyclohexyl-2-[3-(methylsulfanyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N,2-dimethyl-6-(piperidin-3-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]pyrimidin-4-amine
2-ethyl-4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-(propan-2-yl)piperazine
2-({4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridine
2-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-9-oxa-2-azaspiro[5.5]undecane
1-[4-(3,7-dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl)phenyl]-3-(propan-2-yl)urea
3-[1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]benzoic acid
2-(cyclohexylmethyl)-4-(thiophene-2-carbonyl)morpholine
(2E)-3-(4-methoxyphenyl)-1-{4-[5-phenyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}prop-2-en-1-one
1-[2-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-4-fluorophenyl]ethan-1-one
N-{1-[4-(3,4,5-trimethoxyphenyl)phenyl]ethyl}acetamide
8-(quinoxalin-2-yl)-1-oxa-8-azaspiro[4.5]decane
4-methyl-2-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-3-yl}-1H-1,3-benzodiazole
8-chloro-2-{[(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)amino]methyl}quinolin-4-ol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2-(methylamino)-N-(oxolan-2-ylmethyl)acetamide
N-[2-(dimethylamino)ethyl]-N,1-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-3-{[2-(1-phenylethyl)-1H-imidazol-1-yl]methyl}benzamide
methyl 3-[(3S,4R)-1-[(3-methoxyphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
4-hydroxy-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-propyl-1H-pyrazole-4-carboxamide
1-cyclohexyl-4-(3-ethyl-1,2,4-oxadiazol-5-yl)piperidine
6-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-(morpholin-4-yl)pyrimidin-4-amine
2-ethyl-8-[2-(pyrrolidin-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}-4-(pyrrolidin-1-yl)butan-1-one
N-(cyclopropylmethyl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-[(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)formamido]-3-(4-fluorophenyl)propanoic acid
methyl 3-(dimethyl-1,3-thiazole-5-carbonyl)-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl](pyridin-2-ylmethyl)amine
1-methyl-2-({3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
N-[2-(furan-2-yl)ethyl]-6-methoxy-1-methyl-1H-indole-2-carboxamide
2-(4-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}piperidin-1-yl)acetamide
1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidine
3-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}-1,3-oxazolidin-2-one
1-[(6-chloropyridin-3-yl)methyl]-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazine
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-hydroxyphenyl)ethan-1-one
6-ethyl-3-{[(4-hydroxybutan-2-yl)amino]methyl}-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(1R,5R)-6-(cyclopropylmethyl)-3-(6-cyclopropylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-oxo-2-(thiophen-2-yl)acetamide
2-(3-fluorophenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
2-{2-methyl-6-[4-(2-methylpropyl)-1,4-diazepan-1-yl]pyrimidin-4-yl}ethan-1-amine
[(2-methoxyphenyl)methyl]({[8-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl})amine
2-[4-(2-methoxypyridin-3-yl)-1H-pyrazol-1-yl]-N-{1,4,6-trimethyl-1H-pyrazolo[3,4-b]pyridin-3-yl}acetamide
2-(methylamino)-N-[(3R,4S)-4-(propan-2-yl)-1-(3,3,3-trifluoropropyl)pyrrolidin-3-yl]pyrimidine-5-carboxamide
2-(2,4-dichlorophenoxy)-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]acetamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]acetamide