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2-(dimethyl-1,2-oxazol-4-yl)-1-{9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
1-cyclohexyl-3-(cyclopropylmethyl)-N-[(6-hydroxypyrimidin-4-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]-N5-(3-methoxypropyl)piperidine-3,5-dicarboxamide
5-cyclopropanecarbonyl-1'-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(4-chlorophenyl)ethyl]-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-amine
N,N-diethyl-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-{4-[(4-chloro-3-fluorophenyl)methyl]morpholin-3-yl}-N-(cyclopent-3-en-1-yl)acetamide
5-{3-[1-(oxolan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
1-{2-[4-(3-methylbut-2-en-1-yl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
4-(2,3-dihydro-1H-inden-5-yloxy)-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
2-methyl-4-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-1H-1,3-benzodiazole
1-methyl-2-phenyl-4-(1,3-thiazol-2-ylmethyl)piperazine
(2E)-N-{[3-methyl-7-(1H-pyrazole-4-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenylprop-2-enamide
6-(2-methylpropyl)-4-[1-phenyl-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyrimidin-2-one
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-(oxan-4-yl)piperidine-3-carboxamide
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)acetamide
1-(2-benzylmorpholin-4-yl)-3-(4-fluorophenyl)propan-1-one
N-methyl-3-(5-methylfuran-2-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
(1S,5R)-3-cyclobutanecarbonyl-6-(3,5-dimethylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
6-(3,5-dimethoxybenzoyl)-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-[7-(1-benzothiophen-3-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(pyrrolidine-1-carbonyl)piperidine
N-(2-methoxyethyl)-4-[(4-methyl-5-oxo-1,4-diazepan-1-yl)sulfonyl]benzamide
5-[2-chloro-3-(pyrrolidin-1-ylmethyl)phenoxymethyl]-3-(thiophen-2-yl)-1,2,4-oxadiazole
N3-[(4-methylphenyl)methyl]-N5-[3-(methylsulfanyl)propyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
2-(ethylamino)-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}pyrimidine-5-carboxamide
2-[3-(1H-imidazol-1-yl)propyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(2-ethoxyethyl)-N-[(4-fluorophenyl)methyl]-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(1R,5R)-6-[(1-ethyl-1H-indol-4-yl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chloro-2-methylphenyl)urea
2-cyclopentyl-N-cyclopropyl-N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}acetamide
2-[4-(2,5-dimethylfuran-3-carbonyl)piperazin-1-yl]-1,3-benzothiazole
6-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]quinoxaline
N4-[3-(1H-imidazol-1-yl)propyl]-N2,N2,5,6-tetramethylpyrimidine-2,4-diamine
N-(4-methyl-2-oxo-2H-chromen-7-yl)-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
1-[4-(4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one
1-(6-chloro-1,3-benzothiazol-2-yl)-N-(thiolan-3-yl)piperidin-4-amine
N3-[(2-methoxyphenyl)methyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
7-(1,3-benzothiazol-2-yl)-4-(2-ethoxyethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2,5-dimethylphenyl)-3-({[(pyrazin-2-yl)carbamoyl]methyl}amino)propanamide
N-[(2-fluorophenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-(2,4-dimethoxyphenyl)-N-(2-fluorophenyl)furan-2-carboxamide
4-(2,5-dimethoxyphenyl)-2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}phenol
1-butyl-3-cyclopropyl-5-[(3,4-dimethoxyphenyl)methyl]-1H-1,2,4-triazole
3,4,7-trimethyl-2-[4-(pyridin-4-yloxy)piperidine-1-carbonyl]-1H-indole
3-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amine
N-(5-chloro-2-methoxyphenyl)-3-[1-(2-methoxypyridine-3-carbonyl)piperidin-3-yl]propanamide