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3-(4-phenylpiperazine-1-carbonyl)-2,8-diazaspiro[4.5]decane
6-[6-hydroxy-4-(pyridin-4-yl)-1,4-diazepan-1-yl]pyridine-2-carbonitrile
1-methyl-3-(2-methylpropyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
7-(2-phenoxybutanoyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(methylsulfanyl)-N-[1-(pyrazin-2-yl)piperidin-3-yl]acetamide
{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}bis(prop-2-en-1-yl)amine
1-benzyl-N-methyl-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}piperidin-4-amine
N-(1H-indol-2-ylmethyl)-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{2-[2-amino-3-cyano-6-(2-fluorophenyl)pyridin-4-yl]phenoxy}acetic acid
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(3-methylfuran-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(1-{2-[4-(4-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-methylfuran-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(4,5-dimethyl-1H-imidazol-1-yl)acetamide
4-({4-methyl-5-[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-({[2-(methylamino)pyridin-3-yl]methyl}(thiophen-2-ylmethyl)amino)butan-1-ol
1-[3-(furan-2-yl)phenyl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
4-[(1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methyl]morpholine
4-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N,N-dimethyl-4-oxobutanamide
4-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}-1,4-oxazepan-6-ol
N-(2,5-dimethylphenyl)-N'-(prop-2-en-1-yl)-N'-(pyridin-2-ylmethyl)propanediamide
1-(2-propylpyridine-4-carbonyl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
2-methyl-4-(4-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}phenyl)butan-2-ol
5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-methyl-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
4-[(2-methoxyphenyl)methyl]-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
3,5-difluoro-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)pyridine-2-carboxamide
6-(3-ethyl-4-methylpiperazin-1-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
1-(4-chlorophenyl)-N-{[7-fluoro-5-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropane-1-carboxamide
N-(2-{[1-(2-methylpropyl)-6-oxopiperidin-3-yl]formamido}ethyl)pyridine-3-carboxamide
3-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chloro-2-methylphenyl)urea
1-[1-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]-3-phenylpropan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-[1-(furan-2-carbonyl)piperidin-3-yl]-1-(propan-2-yl)-1H-pyrazole-3-carboxamide
9-(2-amino-6-methylpyrimidin-4-yl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[1'-(oxolan-3-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
[(3R,4R)-1-(2,6-dimethylpyrimidine-4-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
4-fluoro-N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
1-[1-(cyclopropylmethyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
1-(3-fluorophenyl)-4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-1H-pyrazole
1-({1-[(4-methylthiophen-2-yl)sulfonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
2-amino-6-cyclopropyl-4-[4-ethoxy-3-(hydroxymethyl)phenyl]pyridine-3-carbonitrile
5-[3-(1H-pyrazol-1-yl)phenyl]-1,2-dihydropyrimidin-2-one
7-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}-4-methyl-2H-chromen-2-one
N-(3-ethoxypyridin-2-yl)-4-[(3-oxopiperazin-1-yl)methyl]benzamide
1-[(3-fluorophenyl)methyl]-4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
N-(1-cycloheptylpiperidin-3-yl)-2-(pyridin-2-yl)acetamide
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-5-methylthiophene-2-carboxamide
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-1H-pyrazole-4-carboxamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-8-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
[(4-{[1-(3-chlorobenzoyl)piperidin-3-yl]methoxy}phenyl)methyl](methyl)(2-phenylethyl)amine
methyl 4-[(3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamido)methyl]benzoate
2-{1-[(2,6-difluoro-4-methoxyphenyl)methyl]piperidin-3-yl}propan-2-ol