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{1-[(2-cyclohexylpyrimidin-5-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
N-[2-(dimethylamino)-1-phenylethyl]-N-methyl-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
(3R,4R)-4-cyclopropyl-1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-3-methylpiperidin-4-ol
2-(2-oxopiperidin-1-yl)-N-{2-[2-(trifluoromethoxy)phenyl]ethyl}acetamide
7-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amine
1-(5-methyl-1,3,4-thiadiazol-2-yl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-2,2-dimethylpropan-1-ol
3-(2-methyl-1-benzofuran-7-yl)-1-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
(1R,5R)-6-[(3,5-dichloropyridin-4-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-{1'-cyclohexanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
3-[(3R,4S)-1-(4-chloro-2-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
4-{5-fluoro-2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidin-4-yl}morpholine
[2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]urea
6-oxo-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1,6-dihydropyridine-3-carboxamide
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyridine-3-carboxamide
1,3-dimethyl 5-{[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]amino}benzene-1,3-dicarboxylate
2-(5-methoxypyridin-3-yl)-N-methylbenzamide
3-phenyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3-phenylpropanamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
4,6-dimethyl-1-[2-(methylsulfanyl)phenyl]piperazin-2-one
N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
N-{2-[2-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}pyridine-3-carboxamide
N-[(5-fluoro-2-methylphenyl)methyl]-2-(4-propanoylphenoxy)acetamide
1-[2-(dimethylamino)ethyl]-4-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]pyrrolidin-2-one
1,3-dimethyl-N-[2-(pyridin-3-yloxy)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2,6-dimethyl-3-(4-methylpiperazine-1-carbonyl)quinoline
N-cyclohexyl-3-({4-[(3-oxopiperazin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine-1-carboxamide
6-butyl-2-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1H-1,2,4-triazole-5-carboxamide
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]pyridine-2-carboxamide
9-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
N3-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}piperidine-1,3-dicarboxamide
1-[5-(cyclopentylamino)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl]piperidin-4-ol
(3S,9aR)-3-(4-aminobutyl)-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(4-chlorophenyl)methyl]-N-(2-hydroxyethyl)-6-oxo-N-propylpiperidine-3-carboxamide
N-[1-(2-phenylethyl)piperidin-4-yl]-4-(pyridin-2-yl)pyrimidin-2-amine
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanamide
1-[(dimethyl-1,2-oxazol-4-yl)carbamoyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-cyclopentyl-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N-{3-[({2-[(pyridin-3-yl)amino]ethyl}carbamoyl)amino]phenyl}cyclopentanecarboxamide
5-(2-fluorophenyl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-({4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
N-methyl-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
1-(3,5-dimethylphenyl)-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperazin-2-one
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}acetamide
(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(prop-2-en-1-yl)piperidin-3-yl)methanol
N-[(3S,4R)-1-(2-methylquinolin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide