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N-[(2,5-dimethylphenyl)methyl]-N-(pyridin-2-ylmethyl)cyclopropanamine
2-(oxolan-2-ylmethyl)-4-[4-(3-phenylpropyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[(3S)-1-benzylpyrrolidin-3-yl]-5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
5-oxo-N-[(1-propyl-1H-imidazol-2-yl)methyl]-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
(2S)-2-[2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]-3-methylbutanamide
ethyl 4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
2-(cyclohex-1-en-1-yl)-1-{4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
1-[2-(pyridin-3-yl)-4-{[2-(1H-pyrrol-1-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-(1-cyclopropylethyl)-5-(2-methoxyphenyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
(1R,9S)-11-[2-(propan-2-yl)-1,3-benzoxazole-5-carbonyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-(2-{[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)acetic acid
3-[(5-hydroxy-4-oxo-4H-pyran-2-yl)formamido]-N-(naphthalen-1-yl)propanamide
10-methoxy-5-(trimethyl-1H-pyrazole-4-carbonyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
(3aS,7aR)-5-methyl-2-[3-(pyridin-3-yl)propanoyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
2-[1-cyclopentyl-4-(2,3-dimethyl-1H-indole-7-carbonyl)piperazin-2-yl]ethan-1-ol
1-(4-{[(1S)-2-hydroxy-1-phenylethyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-(1,2-benzoxazol-3-yl)-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]acetamide
dimethyl[1-(3-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}phenyl)ethyl]amine
(1S,9R)-11-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
N-(butan-2-yl)-2-chloro-4-acetamido-N-(pyridin-3-ylmethyl)benzamide
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-phenylethan-1-one
N-[2-(3-methoxyphenyl)phenyl]-1-(1H-pyrazole-3-carbonyl)piperidine-4-carboxamide
1-ethyl-5-[4-methoxy-3-(methoxymethyl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazole
N-methyl-5-(phenoxymethyl)-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
butyl 4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
4-{1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperidin-4-yl}pyridine
{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
N-[(3,5-dimethoxyphenyl)methyl]-3-(1H-imidazol-2-yl)benzamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2-[2-(2-methoxyethyl)-2H-1,2,3,4-tetrazol-5-yl]morpholine
2-(dimethylamino)-2-(2-fluorophenyl)-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
N-methyl-3-[methyl({[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino]butanamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(2-methylpyrimidin-4-yl)piperazin-2-yl}ethan-1-ol
5-{1-[(2,6-difluorophenyl)methyl]-1H-imidazol-2-yl}-2-(2-methoxyethyl)pyrimidine
5-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]-3-methyl-1H-1,2,4-triazole
4-cyano-N-[(3R,4S)-1-(2-hydroxyethyl)-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
1-(2-benzyl-1,3-thiazole-4-carbonyl)-3-[(dimethylamino)methyl]piperidin-3-ol
1-{3-[4-(benzyloxy)piperidine-1-carbonyl]piperidin-1-yl}propan-1-one
4-[2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)acetyl]-1λ6-thiomorpholine-1,1-dione
2-{[1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
(1R,2R,6S,7S)-4-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-{4-[1-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-imidazol-2-yl]phenyl}acetamide
3-{[3-cyclopropyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
5-(3-fluorophenoxymethyl)-N-(2-hydroxyethyl)-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-phenylacetamide
5-{[benzyl(methyl)amino]methyl}-N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-(1H-indazol-6-yl)-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
3-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-6-methylpyrazolo[1,5-a]pyrimidine
5-(1-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-1H-imidazol-2-yl)-N,N-dimethylpyrimidin-2-amine