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(4aS,8aR)-6-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide
1-[5-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]pyrrolidine
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]acetamide
ethyl N-{[(2S,4S)-4-fluoro-1-(1H-1,2,4-triazole-5-carbonyl)pyrrolidin-2-yl]methyl}carbamate
2-({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
4-(2-methoxyphenyl)-2-methyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperazine
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[3-(morpholin-4-yl)propyl]amine
4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
3-(1H-1,2,3-benzotriazol-4-yl)-1-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
2-[(3,4-dimethylphenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
dimethyl(2-{[(5-methylthiophen-2-yl)methyl]({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl})amino}ethyl)amine
2-cyclohexanecarbonyl-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-methyl-8-{[3-(prop-2-yn-1-yloxy)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1R,5S,6R)-3-[(2,4-diethoxy-3-methylphenyl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
N-[2-({2-oxo-1-oxaspiro[4.4]nonan-4-yl}formamido)ethyl]pyridine-3-carboxamide
1-(2-methylphenyl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,4-diazepane
3-benzyl-5-(4-methoxycyclohexyl)-1H-1,2,4-triazole
5-(3,3-diphenylpiperidine-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
4-{2-[1-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-2-yl]ethyl}morpholine
2-methyl-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}propan-1-one
2-fluoro-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-sulfamoylbenzamide
N-[3-(1H-imidazol-1-yl)propyl]-2,6-dimethylquinoline-4-carboxamide
4-phenyl-3-[1-(pyrrolidine-1-sulfonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 4-({[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)benzoate
N-(1-methoxybutan-2-yl)-5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-(1-{1-[(3-phenoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2-methylprop-2-en-1-yl)piperidine-3-carboxamide
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
N-[2-(N-methylmethanesulfonamido)ethyl]-2-(1H-pyrrol-1-yl)propanamide
N,3,6-trimethyl-N-(propan-2-yl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-(furan-2-yl)-N-methyl-2-oxoacetamide
N-(1-{1-[(4-hydroxy-3,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-1-phenylpiperidin-4-amine
(9aS)-2-[(2R)-oxolane-2-carbonyl]-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
N-(3-ethoxypropyl)-2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
8-(2-methylpyrimidine-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
N-benzyl-N-[(1R,2R)-2-hydroxycyclohexyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-[4-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
3-ethyl-4-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
N-tert-butyl-3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carboxamide
(4aS,8aR)-6-{[4-(pyridin-2-yl)phenyl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
[(2-butyl-1H-imidazol-4-yl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-propyl-1,3-thiazole
2-(4-methylphenyl)-5-[4-(pyridin-3-yl)piperazine-1-carbonyl]pyrimidin-4-ol
1-[7-(1-benzothiophen-3-yl)-9-ethoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}-N-cyclopropylpropanamide