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2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(2-acetamidoethyl)acetamide
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
1-(oxolan-2-ylmethyl)-3-(1-propyl-1H-1,2,3-triazol-4-yl)-1-(thiophen-3-ylmethyl)urea
4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
2-[2-(1H-imidazol-4-yl)ethyl]-9-(5-methyl-1,3-oxazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
7-({[cyclopropyl(pyridin-2-yl)methyl](methyl)amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
9-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3,9-diazaspiro[5.6]dodecane
2-methyl-4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(2-methyl-1H-indol-1-yl)propanamide
[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
3-[(3R,4S)-1-[2-(3-fluorophenyl)acetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(1S,4S)-2-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane
2-(dimethylamino)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-(2-methylphenyl)acetamide
N-ethyl-N-(4-hydroxybutan-2-yl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(4-{[3-(aminomethyl)piperidin-1-yl]methyl}phenyl)-6-(2-methyl-1,3-thiazol-4-yl)-3,4-dihydropyrimidin-4-one
2-methyl-4-[5-({[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amino}methyl)thiophen-2-yl]but-3-yn-2-ol
N'-{[7-chloro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N'-[2-(4-fluorophenyl)ethyl]-N,N-dimethylbutanediamide
2-(4-chlorophenyl)-4-(2-propylpyridine-4-carbonyl)morpholine
1-{2-[4-(3,3-dimethylbutanoyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-[(2-methoxyphenyl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-cyclopropyl-1-{1-[1-(3,4-dimethoxyphenyl)propan-2-yl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
3-(1-phenoxypropan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-{[(1,3-thiazol-2-yl)carbamoyl]methyl}propanamide
7-(cyclopropylmethyl)-N-(2,2-difluoroethyl)-6-(4-methoxyphenyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N,2,4-trimethyl-N-[(4-phenoxyphenyl)methyl]pyrimidine-5-carboxamide
5-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-2,3-dimethylbenzene-1-sulfonamide
1,3-dimethyl-6-[3-(pyridin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(furan-2-ylmethyl)-N-[3-(1H-indazol-1-yl)propyl]piperidine-4-carboxamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(2-methoxyphenoxy)ethan-1-one
1-{4-[4-methoxy-2-(1,4-oxazepane-4-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
2-[N-methyl-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamido]-2-(thiophen-2-yl)acetic acid
2-{3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]phenoxy}acetamide
3-{[(2,2-dimethyloxan-4-yl)(methyl)amino]methyl}benzoic acid
2-(1H-imidazole-5-carbonyl)-6-methyl-5-[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
3-{[1-(cyclohexylmethyl)-1H-1,2,4-triazol-5-yl]methyl}pyridine
(2S,3S)-2-({2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazol-5-yl}formamido)-3-methylpentanamide
N-[(5-methylfuran-2-yl)methyl]-3-[1-(4,4,4-trifluorobutanoyl)piperidin-3-yl]propanamide
N-[(3S,4R)-1-[2-(methylamino)acetyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
(2S,4S)-4-amino-1-{2,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carbonyl}-N-ethylpyrrolidine-2-carboxamide
1-ethyl-3-(2-methylphenyl)-3-[2-(morpholin-4-yl)-2-oxoethyl]pyrrolidine-2,5-dione
1-[(1S,5R)-6-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-methyl-5-(2-methylpropyl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
3-(2-phenylethyl)-8-(piperidin-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-ethyl-8-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(1-ethyl-1H-pyrazole-4-carbonyl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[5-(5-ethyl-1,3,4-oxadiazol-2-yl)-2-methoxyphenyl]-3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]urea
4-(4-phenyl-1H-pyrazol-5-yl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
2-(propylsulfanyl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one