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(4aS,8aR)-1-butyl-6-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,1-dimethyl-5-phenyl-1H-pyrrole-2-carboxamide
4-[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]-6-methyl-2-(pyridin-3-yl)pyrimidine
4-({1-[ethyl(methyl)amino]hex-5-en-2-yl}oxy)-2-methoxypyridine-3-carbonitrile
1-(piperidin-1-yl)-2-[(3S,4R)-3-propyl-4-[(pyrimidin-2-yl)amino]pyrrolidin-1-yl]ethan-1-one
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)acetamide
N3-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)piperidine-1,3-dicarboxamide
N-(1-oxo-1-{4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}pentan-2-yl)acetamide
2-[4-oxo-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]benzonitrile
5-(morpholin-4-yl)-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole
(3S,4S)-1-(1-methanesulfonylpiperidin-4-yl)-4-(3-methoxyphenyl)piperidin-3-ol
1-(4-aminopyrimidin-2-yl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
(3S,4R)-1-(1,3-benzothiazol-2-yl)-3-ethyl-4-methylpiperidin-4-ol
5-chloro-N-[5-methoxy-2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyridine-2-carboxamide
1-methyl-8-(4-methylpyridine-3-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(1-benzothiophene-5-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
4-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]sulfonyl}-2,1,3-benzothiadiazole
2-amino-6-(3-hydroxyphenyl)-4-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
1-methyl-4-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}piperazine
5-(1-ethyl-1H-pyrazol-3-yl)-1-(2-methoxyphenyl)-1H-1,2,4-triazole
3-{2-methyl-2,7-diazaspiro[4.5]decane-7-carbonyl}aniline
3-[(3R,4S)-1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
6-({[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}amino)pyridine-3-carbonitrile
methyl 3-{methyl[1-(3-phenylpropyl)piperidin-3-yl]carbamoyl}benzoate
2-methyl-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-2-(1H-pyrrol-1-yl)propan-1-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-methylpiperidine
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
4-[4-({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)piperidin-1-yl]-N-[(2-fluorophenyl)methyl]benzamide
1-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
3-{[({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)amino]methyl}pyrrolidin-3-ol
3-(2-methoxyethyl)-1-[4-(1H-pyrazol-4-yl)butanoyl]piperidine-3-carboxylic acid
8-(2-cyclopropylacetyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3,5-difluoro-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)pyridine-2-carboxamide
methyl 3-(oxolane-3-amido)-1-(2-phenylethyl)-5-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{[2-cyclopropyl-7-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}acetamide
methyl(2-{4-[3-(2-methylphenyl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)amine
8-[(2-aminopyridin-3-yl)methyl]-2-benzyl-2,8-diazaspiro[5.5]undecan-3-one
2-(3-methoxypropyl)-8-[2-(1H-pyrazol-1-ylmethyl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
(1-benzothiophen-2-ylmethyl)(methyl){[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}amine
4-(hydroxymethyl)-1-[5-(3-methoxyphenyl)furan-2-carbonyl]piperidin-4-ol
15-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-13-oxo-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
8-(2-aminoacetyl)-3-[3-(4-ethylpiperazin-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5R)-3-(5-methylpyrazine-2-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(4-benzoylpiperidin-1-yl)-1-(3-methylpiperidin-1-yl)propan-1-one
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(dimethyl-1,2-oxazol-4-yl)acetamide
(4aR,7aS)-1-methanesulfonyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-fluoro-2-[({[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}amino)methyl]quinolin-4-ol
N-{[3-(dimethylamino)phenyl]methyl}-3-(3-hydroxy-3-methylbutyl)benzamide
methyl 6-{3-[4-(ethoxycarbonyl)piperazin-1-yl]piperidin-1-yl}pyrazine-2-carboxylate