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2-{[1-(4-fluorophenyl)propyl]amino}propane-1,3-diol
(3S,4S)-N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-3-(dimethylamino)-4-hydroxypyrrolidine-1-carboxamide
(2S,4R)-4-hydroxy-N-methyl-N-[(4-phenoxyphenyl)methyl]pyrrolidine-2-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
(1R,5S)-8-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,8-diazabicyclo[3.2.1]octane
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-4-phenylbutan-1-one
(2S,4S)-N-[(4-methylphenyl)methyl]-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
3-fluoro-4-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyridine
methyl 4-{[4-(4-fluorobenzoyl)-7-oxo-1,4-diazepan-1-yl]methyl}benzoate
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
5-cyclopropanecarbonyl-1'-{thieno[2,3-d]pyrimidin-4-yl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
(5S,9aS,9bS)-5-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-4-(pyridin-2-ylmethyl)piperazin-2-one
3-(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)propan-1-ol
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-{2-[(2-methylphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-{thieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
(1R,2R,6S,7S)-4-[(1-methyl-1H-imidazol-2-yl)methyl]-4-azatricyclo[5.2.1.02,6]decane
1-(4-methyl-1,3-thiazole-5-carbonyl)-3-(2-phenylethyl)piperidine
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(prop-2-en-1-yl)acetamide
(3aR,6aR)-2-{[(4-methoxyphenyl)methyl]carbamoyl}-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(3,4-dichlorophenyl)-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazole
1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
1-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(2,3-dihydro-1H-indene-1-carbonyl)piperidine
2-(2,3-difluorophenoxymethyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
N-ethyl-4-methyl-5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,3-thiazol-2-amine
(1S,5R)-6-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)-3-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
1-methyl-8-(2-methylpropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-({8-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1,3-diazinane-2,4-dione
N-butyl-1-ethyl-N-(furan-2-ylmethyl)-7-methyl-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide
3-{[1-(2-methyl-6-propylpyrimidin-4-yl)pyrrolidin-3-yl]methyl}benzamide
3-chloro-N-cyclopentyl-4-{[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]oxy}benzamide
2-[2-(dimethylamino)ethyl]-9-(2,4-dimethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
(3R,4R)-1-{[3-(furan-2-yl)phenyl]methyl}-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]pyrrolidin-3-yl]methanol
N-(3-cyclopentylpropyl)-N-methylthiophene-2-carboxamide
N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-(thiophen-2-ylmethyl)benzamide
3-({[(2E)-3,7-dimethylocta-2,6-dien-1-yl]carbamoyl}amino)benzamide
N-[3-(2-methoxybenzamido)phenyl]-1H-imidazole-2-carboxamide
2-[2-(dimethylamino)ethyl]-9-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
9-(2-ethoxypropanoyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(5-methylpyridin-2-yl)-1-[(2R)-pyrrolidine-2-carbonyl]piperidin-4-ol
N-(5-methyl-1,2-oxazol-3-yl)-2-(4-methyl-1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-[1-(2,4-dimethylphenyl)propyl]-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-(azepan-1-yl)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]acetamide
3-{2-[4-(2,4-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-4-(thiophen-2-ylmethyl)piperazin-2-one