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3-[(4-fluorophenyl)formamido]-N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
{6-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]pyridin-2-yl}methanol
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3,3-dimethylbutan-1-one
2-methyl-5-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyrimidine
2-(2-{1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
2-cyclobutanecarbonyl-7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinoline
1-(4-{[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenyl)ethan-1-one
1-methyl-2-oxo-8-[2-(pyridin-3-yl)acetyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-methyl-1-(4-methylphenyl)-4-[2-(2,3,4-trifluorophenyl)acetyl]piperazin-2-one
dimethyl({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}sulfamoyl)amine
N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-(2-methylfuran-3-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-[(2R)-3-methylbutan-2-yl]urea
1-{2-oxo-2-[3-(pyrrolidin-1-yl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-cyclopropyl-8-(3-hydroxy-2-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{[1-(2-fluorophenyl)propan-2-yl]amino}hexan-1-ol
1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethan-1-amine
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(piperidine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-(5-methylthiophene-2-carbonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]pyrimidin-2-amine
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-[(4-hydroxyphenyl)methyl]-N-(2-methylpropyl)piperidine-3-carboxamide
2-({3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
N-methyl-2-({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)propanamide
1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-4-phenyl-1,4-diazepane
2-{4-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
2-{3-[2-(methylsulfanyl)ethyl]-5-[1-(oxan-4-yl)piperidin-3-yl]-1H-1,2,4-triazol-1-yl}acetic acid
1-[1-(2-phenoxyethyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
1-methyl-2-{5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-1,3-benzodiazole
2,6-dimethoxy-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]pyridine-3-carboxamide
N-[2-(dimethylamino)ethyl]-6-oxo-N-(thiophen-3-ylmethyl)-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-[2-(azepan-1-yl)ethyl]-3,5-diacetamido-N-ethylbenzamide
4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}quinoline
4-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutanamide
N-[(3S,4R)-1-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
6-cyclopentyl-1-methyl-N-(pyridin-2-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-phenylpropan-1-one
2-(morpholin-4-yl)-1-[3-(pyridin-2-yl)azetidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-[(2-fluorophenyl)methyl]-2-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]acetamide
(3S,4R)-4-(pyridin-4-yl)-1-(quinolin-4-ylmethyl)pyrrolidine-3-carboxylic acid
2-[(1S,5R)-3-(1,3-benzothiazole-6-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
ethyl 4-[({[(2-fluorophenyl)methyl]carbamoyl}methyl)amino]piperidine-1-carboxylate
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-1-(furan-2-ylmethyl)piperidine-3-carboxamide
(2S,4R)-4-cyclopropaneamido-N,N-diethyl-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidine-2-carboxamide
N-[(6-chloroquinolin-2-yl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(2-methylphenyl)methyl]piperidine
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}(pentan-2-yl)amine
3-[2-(benzenesulfonyl)ethyl]-4-(hydroxymethyl)-1,3-oxazolidin-2-one
2-methyl-8-(thiophene-3-sulfonyl)-2,8-diazaspiro[4.5]decan-3-one