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2-[(4,5-dimethylfuran-2-yl)methyl]-2,8-diazaspiro[4.5]decane
ethyl 1-[(4-fluoro-3-methoxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-[2-(4-methoxyphenyl)ethyl]-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{3-cyclopentyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-methoxy-4-methyl-1,3-thiazole
5-(oxolan-2-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}thiophene-2-carboxamide
N-cyclobutyl-2-(3-methyl-1H-pyrazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(3aS,6aR)-5-(1-ethyl-1H-pyrazole-4-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(1R,2R,6S,7S)-4-[5-(methanesulfonylmethyl)pyridin-2-yl]-4-azatricyclo[5.2.1.02,6]decane
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-[2-(2-fluorophenyl)ethyl]piperidin-4-amine
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(3-methylbutyl)-1H-pyrazole-3-carboxamide
(1S,5R)-6-(morpholine-4-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-methoxypyridine-3-carboxamide
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-(2-methylphenyl)-1,4-diazepane
(4aS,8aR)-1-(3-methoxypropyl)-6-[3-(1H-pyrazol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
6-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(3-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}butyl)-1H-indole
7-{4-[4-(2-methoxyethyl)phenoxymethyl]phenyl}-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
2-{[4-(cyclopent-3-ene-1-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]methyl}benzoic acid
3-[(2-fluorophenyl)formamido]-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-5-methyl-1,3-oxazole-4-carboxamide
(2R,3R)-3-(dimethylamino)-1'-(3,6-dimethylpyrazin-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(3S)-2-oxoazepan-3-yl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
(3S,4R)-4-(3-fluorophenyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-ol
8-(2,3-dihydro-1H-inden-2-yl)-3-[2-(dimethylamino)ethyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[3-(1H-imidazol-2-yl)phenyl]methyl}(methyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-{3-[(dimethylsulfamoyl)amino]phenyl}urea
4-(1,1-dioxo-1λ6-thiolan-3-yl)-N-[2-(methylsulfanyl)phenyl]piperazine-1-carboxamide
(2S,4R)-4-amino-N-ethyl-1-(4-oxo-1,4-dihydroquinoline-2-carbonyl)pyrrolidine-2-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-N-(3,5-dimethylphenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-cycloheptyl-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-cyclopropyl-3-[2-(3,4-dichlorophenyl)morpholin-4-yl]propanamide
1-(2,3-dihydro-1H-inden-2-yl)-N-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-amine
1-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-3-yl}-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
4,6-dimethyl-2-(2-{4-phenyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}ethyl)pyrimidine
3-[5-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]-1-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}urea
3-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-4-methylphenyl)urea
2-{4-[(5-acetylthiophen-3-yl)methyl]morpholin-3-yl}acetic acid
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(2H-1,3-benzodioxol-5-ylmethyl)(methyl)({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)amine
(3aS,6aR)-3-cyclopentyl-5-(pyrimidin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
7-fluoro-N-(2-methoxyethyl)-3-methyl-N-(1-methylpiperidin-4-yl)-1H-indole-2-carboxamide
methyl (2S,4R)-4-{[(2,5-dimethylphenyl)carbamoyl]amino}-1-methylpyrrolidine-2-carboxylate
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
7-cyclopentyl-2-(5-ethyl-1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(2-chloro-4-fluorophenyl)-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
(1S,5R)-3-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2,6,8-trimethyl-4-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]quinoline
4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-6-methylpyrimidin-2-amine