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6-(2-fluoro-4-methoxyphenyl)-N,7-dimethyl-8-oxo-N-(propan-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-{imidazo[1,2-a]pyridin-3-yl}ethan-1-one
(3R,4R)-1-(benzenesulfonyl)-4-{[2-(1H-imidazol-4-yl)ethyl]amino}pyrrolidin-3-ol
2-(benzyloxy)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-(2,3-difluorophenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyridine-3-sulfonamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[4-(3-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]ethan-1-one
3,3,3-trifluoro-1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
1-(3,4-difluorobenzoyl)-N-(4-fluorophenyl)piperidin-3-amine
1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-4-(pyridin-3-yl)piperazine
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(1-benzylpiperidin-4-yl)methyl]-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
N,2,3,5-tetramethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-(5-{3-[(2-fluorophenyl)formamido]propanoyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
N-cyclopropyl-5-[2-(ethanesulfonyl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-{2-[(2-phenoxyethyl)amino]ethyl}-1-[(4-phenyloxan-4-yl)methyl]pyrrolidin-2-one
6-methyl-2-({1-oxo-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]propan-2-yl}sulfanyl)-3,4-dihydropyrimidin-4-one
N-cyclohexyl-3,5-dimethyl-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
3-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]pyridine
N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
7-methyl-3-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-2,5-dimethylfuran-3-carboxamide
5-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-2-(propan-2-yl)pyrimidine
4-(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)-1-[(2E)-2-methylbut-2-en-1-yl]piperidine
1-{1'-[4-methyl-6-(methylamino)pyrimidin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
2-(4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
4-{2-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]acetamide
(3R,4S)-4-(propan-2-yl)-1-[4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-amine
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
4-cyclopropyl-6-(3,4,5-trimethoxyphenyl)pyrimidine
3-{[(1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-(pyridin-2-ylsulfanyl)propan-1-one
N-(3-hydroxypropyl)-1-{1-[(2-methoxynaphthalen-1-yl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
2-{4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]morpholin-3-yl}acetic acid
2-(2,2-dimethylpropanoyl)-N-[(5-methylfuran-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1'-[3-(1H-imidazol-2-yl)benzoyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-benzyl-N-methyl-3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzamide
(2S,4R)-N-methyl-4-{[(4-phenylphenyl)methyl]amino}-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
1-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}urea
7-(cyclohexylmethyl)-2-[3-(methylsulfanyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-[2-(4-fluorophenyl)ethyl]-4-[4-(2-oxo-2H-chromene-3-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
5-butyl-1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazole
N-[3-(1H-imidazol-1-yl)propyl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
2-cyclopentyl-N-(4-ethoxyphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-(2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)-N-methylacetamide
5-amino-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-phenyl-1H-pyrazole-3-carboxamide
8-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
6-methyl-4-[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
{7-chloro-5-[2-(piperazin-1-yl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine