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3-[(dimethylamino)methyl]-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-3-ol
N-cyclooctyl-4-oxo-4-(3-oxo-4-phenylpiperazin-1-yl)butanamide
(1R,2S,9R)-11-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
5-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-2-methylphenol
2-[(4aR,7aS)-4-{imidazo[1,2-a]pyridin-2-ylmethyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2-{[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]methyl}benzoic acid
1-(5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophen-2-yl)ethan-1-one
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-5-methyl-3,4-dihydroquinazolin-4-one
(3R,5S)-1-benzyl-N3-(4-fluorophenyl)-N5-(2-phenoxyethyl)piperidine-3,5-dicarboxamide
3-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}methyl)pyridin-2-amine
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-methyl-N-(2-phenoxyethyl)acetamide
4-[2-(1H-imidazol-2-yl)benzoyl]-1-(4-methoxyphenyl)-2,2-dimethylpiperazine
N-(1-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-cyclopropylpyridine-2-carboxamide
methyl 5-{[(3-fluorophenyl)methyl]amino}-3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-methyl-4-(5-methylpyrimidin-2-yl)-1,4,9-triazaspiro[5.5]undecane
2-amino-4-{[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]amino}quinazoline-6-carboxylic acid
methyl (2S,4R)-1-methyl-4-[2-(pyridin-3-yloxy)acetamido]pyrrolidine-2-carboxylate
N-[(3S,5S)-5-[ethyl(pyridin-4-ylmethyl)carbamoyl]-1-methylpyrrolidin-3-yl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-({2-[3-(1H-pyrazol-1-yl)phenyl]phenyl}methyl)propanamide
N,N,2-triethyl-6-methyl-4-oxo-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-4-sulfamoylbenzamide
1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
(3R,5S)-N3-methyl-N3-[(3-methylpyridin-2-yl)methyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
2-(3-phenylpiperidin-1-yl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
[4-({1-[(2,6-dimethoxyphenyl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
3-[(dimethylamino)methyl]-1-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}piperidin-3-ol
5-(methoxymethyl)-N-methyl-N-(3-phenylpropyl)-1,3,4-oxadiazole-2-carboxamide
(3S,9aR)-3-benzyl-8-(3-phenylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-({3-[3-(pyrrolidin-1-yl)pyrazin-2-yl]phenyl}methyl)morpholine
6-(benzyloxy)-4-[(3-methylquinoxalin-2-yl)methyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-[1-(2,6-dimethylphenoxy)propan-2-yl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
6-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}pyrazine-2-carboxamide
(benzylsulfamoyl)[2-phenyl-2-(piperidin-1-yl)ethyl]amine
(3S,4R)-1-[2-(2-ethoxyethoxy)benzoyl]-4-methylpiperidine-3,4-diol
4-(1H-1,3-benzodiazol-1-yl)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidine-4-carboxylic acid
7-methoxy-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1,2,3,4-tetrahydronaphthalen-2-amine
1-(3-chlorophenyl)-4-[1-(1H-pyrazol-3-ylmethyl)piperidin-3-yl]piperazine
4-[3-(2-methylphenyl)piperidine-1-carbonyl]benzene-1-sulfonamide
2-{[3-(3-hydroxy-3-methylbutyl)phenyl]formamido}-N,N-dimethylacetamide
4-{2-[2-(ethoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-7-methyl-3,4-dihydro-2H-1,4-benzothiazin-3-one
2-methoxy-6-({methyl[1-(pyridin-3-yl)propyl]amino}methyl)phenol
dimethyl({[4-methyl-5-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,6-dichlorobenzamide
N-[1-(methoxymethyl)cyclopentyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
3-(diphenylmethyl)-N-(thiophen-3-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4-(methylsulfanyl)benzamide
2-(1-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-amine
1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one