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N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-2-(propylsulfanyl)acetamide
1-[1-(2,3,5,6-tetramethylbenzoyl)azetidin-3-yl]piperidine
2-ethyl-9-[2-(4-fluoro-3-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-methyl-N-[2-(morpholin-4-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(1S,6R)-3-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
2-oxo-N-(pyridin-4-ylmethyl)-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(1R,2S,3S,4R,5S)-N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]tricyclo[3.2.1.02,4]octane-3-carboxamide
4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-1,9-dioxaspiro[5.5]undecan-4-amine
{[5-(4-methanesulfonylphenyl)-2-methoxyphenyl]methyl}(methyl)amine
3-(2-hydroxyphenyl)-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1H-pyrazole-5-carboxamide
2-(adamantan-1-yl)-N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}acetamide
1-{1H-pyrrolo[2,3-b]pyridin-6-yl}-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
1-(furan-2-ylmethyl)-4-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidine
3-{[cyclopropyl(2-methylpropyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-methoxy-N-(3-{4-[2-(pyridin-2-yl)piperidin-1-yl]piperidin-1-yl}phenyl)benzamide
2-(2,3-dihydro-1H-indol-1-yl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
{1-[1-(3-fluoro-4-methylbenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}(phenyl)methanol
3-(4-methoxyphenyl)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
3-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-4-amine
4-{5-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazol-5-yl]-1-ethyl-1H-1,2,4-triazol-3-yl}benzamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
7-(cyclohexylmethyl)-2-[(1-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2,6-dimethylbenzamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-3-methylpiperidine
1-(5-phenyl-1,2-oxazole-3-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-(2-methoxyethoxy)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
5-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
ethyl 4-benzyl-1-[(5-acetamidoquinolin-2-yl)methyl]piperidine-4-carboxylate
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
[(2-methyl-1H-imidazol-4-yl)methyl](oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
N-cyclopentyl-5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2-methoxy-5-{[4-(propan-2-yl)piperazin-1-yl]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
14-(3,5-dichlorophenyl)-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
({2-[(2-chlorophenyl)methoxy]-7-methoxyquinolin-3-yl}methyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
N-{[3-(difluoromethoxy)phenyl]methyl}-3-(1H-pyrazol-1-yl)benzamide
(1S,3R)-N1-[2-(2-ethoxyphenyl)ethyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}urea
1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-5-[2-(prop-2-en-1-yloxy)phenyl]-1H-imidazole
2-(2-{1-[3-(1H-pyrrol-1-yl)propyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
1-methyl-5-[methyl(2-methylpropyl)amino]-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-cyclopropyl-8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
5-(4-fluoro-3-methylphenoxymethyl)-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
N-(1-benzothiophen-2-ylmethyl)-N-methyl-3-(3-methylpiperidin-1-yl)propanamide
1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-[2-(piperidin-1-yl)ethyl]piperidine-4-carboxamide
3-(3-methoxyphenyl)-5-[4-(methylsulfanyl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine