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(1R,2S,6R,7S)-4-[(2-ethylpyrimidin-4-yl)methyl]-4-azatricyclo[5.2.2.02,6]undecane
1-(4-{[2-(dimethylamino)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
(3aS,6aS)-5-[(3-chloro-4-fluorophenyl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-ol
N-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
2-oxo-N-(propan-2-yl)-2-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}acetamide
3-(1-benzyl-1H-imidazol-2-yl)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidine
1-(4-fluoro-2-methylbenzoyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-({1-[2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})(oxan-4-ylmethyl)amine
4-methoxy-N-methyl-3-[3-(1H-pyrazol-3-yl)phenyl]benzamide
benzyl (1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
4-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
(1r,4r)-4-(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidine-1-carbonyl)cyclohexan-1-ol
4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]-1-[3-(trifluoromethyl)benzenesulfonyl]piperidine
2-(3-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}phenoxy)acetamide
N-(5-acetamido-2-methylphenyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carboxamide
3-{[(furan-2-ylmethyl)(methyl)amino]methyl}-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
N-(2-fluorophenyl)-3-{1-[1-(2-methylphenyl)piperidin-4-yl]piperidin-3-yl}propanamide
3-hydroxy-3-({[2-(piperidin-1-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
5-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-2-(2-phenylethyl)-1,3-benzoxazole
4-{4-[1-(dimethylamino)ethyl]piperidin-1-yl}-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
N-[2-(dimethylsulfamoyl)ethyl]-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
8-[4-(methylsulfanyl)benzenesulfonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-benzyl-1-methyl-3-{1-[(2R)-5-oxopyrrolidine-2-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-{5-[(2E)-3-phenylprop-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(propan-2-yl)propanamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(4-formylbenzoyl)piperidine-3-carboxylate
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
3-[4-(3-methylpyridin-4-yl)piperazin-1-yl]propane-1,2-diol
(2R,6R)-4-[(2-aminopyridin-3-yl)methyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(3R,5R)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(pyrrolidin-1-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidine
2-methyl-6-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}phenol
5,7-dimethyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrido[2,3-d]pyrimidin-4-amine
(3aS,6aR)-5-(3-chloropyridin-2-yl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[3-({[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
N-[(3R,4S)-4-cyclopropyl-1-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]pyrrolidin-3-yl]-3-ethoxypropanamide
1-{2-[({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)amino]ethyl}piperidin-3-ol
4-(3,5-dichloro-4-methylbenzoyl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
5-{2-oxo-2-[2-oxo-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2,2-dimethyl-N-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]propanamide
(3S,9aR)-8-(4-chlorobenzoyl)-3-[(1R)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methyl-6-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}-1,3-benzothiazole
3-(2-phenylethyl)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
3-[(3R,4S)-4-(dimethylamino)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl]propanoic acid
4-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
8-fluoro-2-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]quinoline
2-(benzyloxy)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one