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3-(2-amino-1,3-thiazol-4-yl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]propanamide
5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}-N-(thiophen-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
1-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-3-[3-(piperidine-1-carbonyl)phenyl]urea
(3R,4S)-4-{4-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-diazepan-1-yl}oxolan-3-ol
1'-[(2,3-dimethyl-1H-indol-7-yl)methyl]-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-ethyl-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(3,5-difluorophenyl)methyl]-8-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
(benzylsulfamoyl)[(1,5-dimethyl-1H-indazol-3-yl)methyl]amine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-3-(pyridin-3-yl)propanamide
1-[(2-chloro-6-fluorophenyl)methyl]-1-cyclopropyl-3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)urea
3-[4-(1-methoxyethyl)phenyl]-5-[(propan-2-yl)sulfamoyl]benzoic acid
2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxamide
3-(2-fluorophenoxymethyl)-1-[3-(1H-imidazol-2-yl)benzoyl]piperidine
N-methyl-4-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane-8-carbonyl}-1,3-thiazol-2-amine
4-[1-(2-methoxypyridine-4-carbonyl)piperidin-3-yl]-2-methyl-6-(pyrrolidin-1-yl)pyrimidine
2-[3-(2,5-dimethylphenyl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-indazol-3-yl)acetamide
4-(4-methyl-1H-pyrazol-1-yl)-1-(thiophene-2-sulfonyl)piperidine-4-carboxylic acid
(1S,5R)-N,N-dimethyl-6-(pyridine-3-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[5-(8-methoxyquinolin-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-(3-oxo-3-{spiro[indene-1,4'-piperidine]-1'-yl}propyl)pyrrolidin-2-one
4-(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidin-1-yl)-6-methylpyrimidin-2-amine
1-[2-(1,1-dioxo-1λ6-thiolan-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]benzamide
5-(methoxymethyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]thiophene-2-carboxamide
3,5-dimethyl-N-[(5-methylthiophen-2-yl)methyl]-4-oxo-N-(prop-2-en-1-yl)-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-[(1-benzylpiperidin-4-yl)amino]-1-[(3-chlorophenyl)methyl]pyrrolidine-2-carboxamide
5-(1-{[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-1,3,4-thiadiazol-2-amine
(3R,4R)-4-cyclobutyl-1-{[4-(2-hydroxyethoxy)phenyl]methyl}-3-methylpiperidin-4-ol
3-[(5-chlorothiophen-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[5-cyclopropyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]quinoxaline
(3aS,6aS)-5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-N,N-dimethyl-octahydropyrrolo[3,4-b]pyrrole-1-carboxamide
1'-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-{[4-(5-fluoro-2-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-(propan-2-yl)pyrimidine
1,9-dimethyl-4-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(3S,4R)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)-4-propylpyrrolidin-3-yl]methanesulfonamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-ethylphenyl)methyl]piperidine
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-({[(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)carbamoyl]amino}methyl)-N,N-dimethylfuran-2-carboxamide
(2S)-2-{5-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}propanamide
1-methyl-4-({1-[3-(trifluoromethyl)benzoyl]piperidin-3-yl}methyl)piperazine
4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
1-(3-chloro-4-methoxyphenyl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-oxopyrrolidine-3-carboxamide
7-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-3-methyl-3,4-dihydroquinazolin-4-one
(4aS,7aR)-1-[2-(propan-2-yl)pyrimidine-4-carbonyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-oxopentanamide
5-methyl-1-(2-methylphenyl)-4-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]piperazin-2-one
4-(2-methyl-1H-imidazol-1-yl)-1-(pyrrolidine-1-carbonyl)piperidine-4-carboxylic acid
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-(dimethylamino)-N-methylbenzamide