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1-(isoquinoline-1-carbonyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
1-ethyl-7-methyl-N-(2-methylpropyl)-4-oxo-N-(pyridin-2-ylmethyl)-1,4-dihydro-1,8-naphthyridine-3-carboxamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-3-yl]acetamide
N-[(2R,3R)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1-methylpiperidin-3-yl)propan-1-one
N-(4-{[2-(2-hydroxyethoxy)ethyl]carbamoyl}phenyl)-2-methylfuran-3-carboxamide
2-[({5-[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)(methyl)amino]acetamide
(2S)-2-({[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl}amino)propanamide
N-cyclopropyl-N-[(4-hydroxy-3-methoxyphenyl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
6-{4-[2-(4-{[(1-benzothiophen-2-ylmethyl)(methyl)amino]methyl}phenoxy)ethyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl[(1-methyl-1H-imidazol-2-yl)methyl]{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
N,N-diethyl-2-{4-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]-1H-1,2,3-triazol-1-yl}acetamide
4,4-difluoro-1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidine
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(3-methoxyphenyl)propanamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanamide
1-methyl-4-[2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{5-[3-(methylsulfanyl)phenyl]furan-2-carbonyl}pyrrolidine
2-{4-methyl-6-[3-(morpholin-4-yl)piperidin-1-yl]pyrimidin-2-yl}phenol
1-(furan-3-carbonyl)-4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1,4-diazepane
1-[(1-{6-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]pyrimidine-5-carboxamide
8-(2,3-dihydro-1H-inden-2-yl)-3-ethyl-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aR,7aS)-1-benzyl-4-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[2-(aminomethyl)-1H,2H-naphtho[2,1-b]furan-7-yl]-N-cyclopropylpyridine-4-carboxamide
6-{1-[(8-methoxyquinolin-2-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
5-{3-[1-(dimethylamino)ethyl]phenyl}pyrimidin-2-amine
1-[(4-fluorophenyl)methyl]-4-{[(4-hydroxyquinolin-2-yl)methyl]amino}pyrrolidin-2-one
N-[(2R)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-oxobutan-2-yl]acetamide
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(8-methoxyquinolin-5-yl)methyl]methylamine
3-{5-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}-2-[4-(pyrimidin-5-yl)-1H-pyrazol-1-yl]acetamide
3-[1-(2-methylphenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]piperidine-1-carboxamide
1-({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)azepan-4-amine
3-{4-[1-(dimethylamino)ethyl]phenyl}-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
ethyl 1-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamido]cyclobutane-1-carboxylate
1-cyclobutanecarbonyl-4-(4-fluorophenyl)-1,4-diazepane
4-{3-[4-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]propyl}morpholine
N,N-diethyl-1-(5-ethyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-amine
N-({7-[(2,5-difluorophenyl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
N-cyclopropyl-4-methoxy-3-{[1-(oxolane-3-carbonyl)piperidin-4-yl]oxy}benzamide
(3R,4S)-1-(3-chloro-4-methylbenzoyl)-4-cyclopropylpyrrolidin-3-amine
(3aS,6aS)-2-(1H-imidazol-4-ylmethyl)-5-[3-(pyridin-3-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2,3-dihydro-1H-inden-2-yl)-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
2-amino-4-(2-aminopyrimidin-5-yl)-6-(3,4-difluorophenyl)pyridine-3-carbonitrile
N-(1-methoxybutan-2-yl)-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}butanamide
1-methyl-6-oxo-N-[(3R,5S)-1-(pent-2-yn-1-yl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-1,6-dihydropyridine-3-carboxamide