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2-hydroxy-N-{imidazo[1,2-a]pyrazin-3-ylmethyl}-4-(methylsulfanyl)butanamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-ethyl-5-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}piperidin-2-one
4-phenyl-3-({1-[3-(pyridin-3-yl)propanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxybenzamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-2-(2-methylpiperidin-1-yl)acetamide
methyl 1-{2-hydroxy-3-[3-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]propyl}piperidine-4-carboxylate
1-[2-fluoro-3-(trifluoromethyl)phenyl]-3-[2-(2-methylpropanesulfonyl)ethyl]urea
1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(4-fluorophenyl)methyl]-5-[(2S)-oxolane-2-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-[3-(morpholin-4-yl)propyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
1-methyl-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
1-(2-amino-9H-purin-6-yl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
1-(2-hydroxyethyl)-5-[(2S)-2-methoxy-2-phenylacetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
5-(1-benzothiophen-3-yl)pyridine-2-carbonitrile
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-[2-(1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)ethyl]acetamide
5-methyl-N-(propan-2-yl)-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-butyl-N-methyl-3-({methyl[(1-methylpiperidin-2-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carboxamide
3-(piperidine-1-carbonyl)-N-propyl-N-(thiophen-3-ylmethyl)pyrazine-2-carboxamide
2-(2,4,5-trimethylbenzoyl)-2,7-diazaspiro[4.5]decane
2-(2,5-dimethylphenoxy)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}propanamide
(3R,4R)-3-cyclopropyl-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-4-methylpyrrolidin-3-ol
1-(1-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)propan-1-ol
1-(6-carbamoylpyrazin-2-yl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-cycloheptyl-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-1H-1,2,3-triazole-4-carboxamide
3-{2-[2-(4-methylpentyl)morpholin-4-yl]-2-oxoethyl}-1,2,3-oxadiazol-3-ium-5-olate
2-methoxy-N-{3-[2-(pyrrolidin-1-yl)acetamido]phenyl}benzamide
6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purin-2-amine
N-methyl-1,1-dioxo-N-(quinolin-5-ylmethyl)-1λ6-thiane-4-carboxamide
2-(4-carbamoylpiperidin-1-yl)-2-{4-[(dimethylcarbamoyl)amino]phenyl}acetic acid
N-[(1-propyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-fluoro-N-[1-(pyridin-3-yl)propan-2-yl]quinazolin-4-amine
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
3-(5-methyl-1H-pyrazol-1-yl)-N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)propanamide
3-chloro-4-fluoro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]benzamide
(2S)-1-[3-(2-methyl-1H-indol-1-yl)propanoyl]pyrrolidine-2-carboxamide
4-hydroxy-4-(1H-imidazol-1-ylmethyl)-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)piperidine-1-carboxamide
3,6-dimethyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1-benzofuran-2-carboxamide
N'-(3,5-dimethylphenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]propanediamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-[(6-methylpyridin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-amino-8-{3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
(1R,3S)-7-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-3-ethoxy-7-azaspiro[3.5]nonan-1-ol
N-({1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-3-yl}methyl)methanesulfonamide
(1S,5R)-6-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-1-ethyl-1H-pyrazole