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2-[methyl(pyridin-3-ylmethyl)amino]-1-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]ethan-1-one
1-{4-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidin-1-yl}ethan-1-one
5-{1-[(3E)-hex-3-enoyl]pyrrolidin-2-yl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]thiophene-2-carboxamide
methyl 6-{2-azabicyclo[2.2.1]hept-5-en-2-ylmethyl}-3-(2-methylbenzamido)thieno[2,3-b]pyridine-2-carboxylate
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-3-methoxypropanamide
2-[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-[2-(4-fluorophenyl)ethyl]acetamide
3,6-dimethyl-4-(4-methyl-1,4-diazepane-1-carbonyl)-2-(1-methyl-1H-pyrazol-4-yl)quinoline
2-cyclopropyl-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]quinoline-4-carboxamide
(3S,4S)-1-{[2-(furan-2-yl)phenyl]methyl}-4-methylpiperidine-3,4-diol
N-{1-[3-(2-ethylphenoxy)azetidin-1-yl]-1-oxopropan-2-yl}methanesulfonamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(4-methylphenyl)propan-1-one
3-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]quinoline
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-{imidazo[1,2-a]pyridin-3-ylmethyl}urea
4-{1-[(3-phenoxyphenyl)methyl]azetidin-3-yl}morpholine
5-{[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-N-propylpyrimidin-2-amine
3-(2H-1,3-benzodioxol-5-yl)-5-(2,3-dihydro-1-benzofuran-7-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-({4-[1-(propane-1-sulfonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
4-cyclobutaneamido-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]benzamide
2-[(1S,5R)-6-[3-(4-chlorophenyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
3-(4-chloro-3-methylphenyl)-1-{[(1r,4r)-4-(hydroxymethyl)cyclohexyl]methyl}urea
4-(1,2-oxazinane-2-carbonyl)-6-(propan-2-yl)pyrimidin-2-amine
2-(8-methylquinolin-5-yl)pyridine-3-carbonitrile
1-[2-(pyrrolidine-1-sulfonyl)ethyl]-3-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]urea
12-[3-hydroxy-3-(hydroxymethyl)piperidine-1-carbonyl]-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
N3-methyl-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-N3-(quinolin-5-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-4-{3-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]phenyl}butan-2-ol
8-(2-hydroxy-4-methylbenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-propyl-5-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyrimidine
{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(trifluoromethyl)phenyl]methyl}amine
4-(1,3-benzoxazol-2-yl)-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
4-(4-amino-5-methylpyrimidin-2-yl)-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{[1-(carbamoylmethyl)piperidin-4-yl]formamido}-3-(4-fluorophenyl)propanoic acid
1'-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]spiro[indene-1,4'-piperidine]
1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-4-yl)ethan-1-one
(1R,9S)-5-amino-12-methyl-3-[2-(1H-pyrazol-1-ylmethyl)phenyl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
4-[5-(ethanesulfonyl)thiophen-2-yl]-1-methyl-1H-pyrrolo[2,3-b]pyridine
N-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
N-(1,4-oxazepan-6-ylmethyl)-1,3-benzoxazol-2-amine
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-N-[3-(methylcarbamoyl)phenyl]piperidine-1-carboxamide
N-(3-hydroxypropyl)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidine-3-carboxamide
3-{3-[2-(3,4-dihydroxyphenyl)-1H-imidazol-1-yl]phenyl}propanoic acid
N-[2-(cyclohexylsulfanyl)ethyl]-1-(3-hydroxyphenyl)-5-oxopyrrolidine-3-carboxamide
4-[(dimethylamino)methyl]-1-(3-methylfuran-2-carbonyl)azepan-4-ol
{3-[(5-methylfuran-2-yl)methyl]-9-[3-(methylsulfanyl)propyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
3-(2,3-dihydro-1H-inden-2-yl)-5-(piperidin-4-yl)-5-propylimidazolidine-2,4-dione
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}pyridine-2-carboxamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(2-methyl-1H-imidazol-1-yl)propanamide
1-(3-methylpyridin-2-yl)-4-[1-(oxan-4-yl)piperidine-4-carbonyl]piperazine
2-amino-4-[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
4-({2-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine