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(1R,3S)-7-(1,3-benzothiazole-6-carbonyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
8-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(4-phenyl-1,3-thiazol-2-yl)piperidine
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
4-(2-methoxyphenyl)-2-methyl-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazine
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amine
(1-{[1-(2-chloro-6-methylbenzenesulfonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanamine
N-(dimethyl-1,2-oxazol-4-yl)-4-[2,5-dioxo-4-(pyridin-3-yl)imidazolidin-4-yl]piperidine-1-carboxamide
2-amino-6-(furan-2-yl)-4-(3,4,5-trimethoxyphenyl)pyridine-3-carbonitrile
1-[2-(1H-pyrazol-1-yl)acetyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-3-(pyrazin-2-yl)propanamide
1-[3-(3-methoxyphenoxy)azetidin-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
ethyl 2-(4-{[4-(3-hydroxyphenyl)piperazine-1-carbonyl]amino}phenyl)acetate
N-cyclopropyl-1-[5-(3-methoxyphenyl)furan-2-carbonyl]piperazine-2-carboxamide
4-({2-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[(4-methoxyphenyl)methyl]-N-(2-methylpropyl)-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
4-[3-(diethylamino)pyrrolidin-1-yl]pyrimidine-5-carboxylic acid
(3S,4S)-1-(furan-2-carbonyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrrolidin-3-ol
N-[(3-fluorophenyl)methyl]-5-methyl-6-(3-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
(2S,4S)-4-amino-N,N-diethyl-1-[2-(4-methoxy-3-methylphenyl)acetyl]pyrrolidine-2-carboxamide
(4aS,7aR)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}pent-4-en-1-one
N-cyclohexyl-2-(4,5-dimethyl-2-oxo-2,3-dihydro-1,3-oxazol-3-yl)-N-methylacetamide
N-({5-[3-(methylsulfanyl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
N-methyl-2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(1H-imidazol-1-yl)butan-2-yl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]pyridin-2-amine
methyl 3-(cyclobutylmethoxy)-5-[(1-methyl-2-oxopyrrolidin-3-yl)carbamoyl]benzoate
2-{4-methoxy-3-[(E)-2-phenylethenyl]phenyl}ethan-1-amine
1,3-dimethyl-4-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(3-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}phenyl)ethan-1-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
N,1-dimethyl-5-phenyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrrole-2-carboxamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-(azocan-1-yl)-N-(2-methoxyethyl)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
2-[1-(2-amino-4-phenylpyrimidine-5-carbonyl)pyrrolidin-3-yl]benzoic acid
1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}-3-phenoxypropan-1-one
methyl 4-{[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-1H-pyrazole-3-carboxylate
1-{2-amino-4-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1H-1,3-benzodiazol-1-yl)propan-1-one
1-(3-methoxybenzoyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
(3aR,6aR)-2-(3-fluoro-4-methoxybenzenesulfonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-ethyl-N,N-dimethylpyrimidin-2-amine
1'-(5-propyl-1,2-oxazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(4aR,7aS)-1-(3-methylbutanoyl)-4-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-[(3-fluorophenyl)methyl]piperidin-2-one
5-[2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxamide