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4-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-1λ6-thiomorpholine-1,1-dione
(1R,7S)-3-(pentan-3-yl)-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-(1-{[4-(hydroxymethyl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
2-[(4aR,7aS)-4-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
9-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(5-acetamido-2-fluorophenyl)-2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-1-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propan-1-one
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl](methyl)(thiophen-2-ylmethyl)amine
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
(3S,9aR)-8-(4-chlorobenzoyl)-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-({4-methyl-5-[1-(4-methylpent-3-en-1-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-4-(4H-1,2,4-triazol-4-yl)benzamide
1-(4-fluorophenyl)-4-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)butane-1,4-dione
5-(azepan-1-yl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
4-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
{2-ethoxy-5-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)methyl]phenyl}methanol
2-{5-cyclopropyl-4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(3-methoxyphenyl)pyrimidine
(1R,5R)-6-benzyl-3-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(2-fluorophenyl)methyl]-5-methyl-2-(2-methylpropanamido)benzamide
4-methyl-2-{1-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
2-amino-4-(2-butyl-1H-imidazol-4-yl)-5-methyl-6-(pyridin-2-yl)pyridine-3-carbonitrile
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)pyrimidin-4-amine
3-(2-phenylethyl)-4-(propan-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(4-hydroxyphenyl)methyl]-3-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
4-({2-[1-(2-fluoro-6-methoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
1-cyclohexyl-3-(1-methyl-1H-1,3-benzodiazol-6-yl)-1-(pyridin-2-ylmethyl)urea
5-methyl-4-{2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-pyrazol-3-one
1-(2-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}ethyl)pyrrolidin-2-one
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-3-methylfuran-2-carboxamide
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
1-(2-chloro-6-methylphenyl)-3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-methylurea
N-cyclopentyl-6-{octahydropyrrolo[1,2-a]piperazin-2-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-[5-({[(3-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[benzyl(methyl)amino]-3-(4-{[(3-methoxypropyl)amino]methyl}phenoxy)propan-2-ol
1-(1H-imidazol-4-ylmethyl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(2S,4S)-4-amino-1-[3-(1H-pyrazol-1-yl)propanoyl]pyrrolidine-2-carboxylic acid
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-[2-(pyridin-2-ylsulfanyl)ethyl]cyclopentane-1,3-dicarboxamide
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]naphthalene-1-carboxamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
(1S,5R)-6-benzyl-3-[2-(2-methoxyethoxy)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)ethyl]acetamide
2-[(3-methoxyphenyl)methyl]-4-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]morpholine
(3R,4S)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-N,N-dimethyl-4-propylpyrrolidin-3-amine
2-[(2-methoxyethyl)(methyl)amino]-N-[(3R,4S)-4-(propan-2-yl)-1-(1,3-thiazol-2-yl)pyrrolidin-3-yl]acetamide
9-ethyl-1-methyl-4-phenylmethanesulfonyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[2-methoxy-4-(morpholin-4-ylmethyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
N-{1-[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-1-oxopentan-2-yl}acetamide
4-{1-[(furan-2-ylmethyl)carbamoyl]piperidin-3-yl}benzoic acid