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2-(prop-2-en-1-yl)-4-{1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-imidazol-2-yl}phenol
1-(azepan-1-yl)-3-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propan-2-ol
2-(1H-indol-3-yl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-(2-cyclopropylpyrimidin-5-yl)-7-methyl-4-(pyrrolidine-1-carbonyl)quinoline
[4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl](phenyl)methanol
3-{2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)-3-(2-methylphenyl)pyrrolidine-2,5-dione
2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(pyridin-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-{[1-(dimethoxy-1,3,5-triazin-2-yl)piperidin-4-yl]methyl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
1-methyl-1-{[3-(thiophen-2-ylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}urea
methyl[(4-propyl-4H-1,2,4-triazol-3-yl)methyl](quinolin-4-ylmethyl)amine
N-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
(5-{[methyl(thian-4-yl)amino]methyl}-2-(propan-2-yloxy)phenyl)methanol
N'-(3-ethylphenyl)-N-[4-(oxolan-2-yl)butyl]butanediamide
3-(oxolan-3-yl)-5-[1-(propan-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazole
1-methyl-3-(thiomorpholine-4-carbonyl)-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyrimidin-4-amine
1-[2-(dimethylamino)-4-{[2-(thiophen-2-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
5-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1H-indole-2-carboxamide
N-[2-(4-methylmorpholin-2-yl)ethyl]-3-(1,2-oxazinan-2-yl)propanamide
(4aR,7aS)-1-propanoyl-4-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[4-methyl-5-(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methanol
5-phenyl-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-5-fluoro-4-(morpholin-4-yl)pyrimidin-2-amine
(3aS,6aR)-5-(1,3-benzothiazol-2-yl)-3-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(1-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
1,3-dimethyl-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(3-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-(3-methoxyphenyl)-5-(oxolan-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-(2-{1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}ethyl)acetamide
1-methyl-3-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]imidazolidine-2,4-dione
3-({1-[3-(2-oxopiperidin-1-yl)propanoyl]pyrrolidin-3-yl}methyl)benzamide
(1R,5R)-6-benzyl-3-(trimethyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-chloro-2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-(2-fluoroethyl)-2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
1-(5-chloropyridin-2-yl)-4-[(2-fluoro-4-methoxyphenyl)methyl]piperazine
(1s,4s)-4-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carbonyl}cyclohexan-1-ol
4-[1-(6-aminopyridine-3-carbonyl)piperidin-4-yl]pyrimidin-2-amine
2-methyl-5-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,3-benzodiazole
2-{4-[(2,3-difluoro-6-methoxyphenyl)methyl]morpholin-2-yl}ethan-1-ol
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-ethyl-5-(methoxymethyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-cyclopentylacetamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(2-methoxypyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-oxo-8-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-6-methylquinoline
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
[(3R,4S)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol