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3-methyl-7-(3-phenoxypropanoyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)piperidine
4-{2-[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]ethyl}phenol
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
[(5-fluoro-1H-indol-2-yl)methyl](methyl){[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
(3S,4S)-4-cyclopropyl-1-[2-(2,4-difluorophenyl)acetyl]pyrrolidine-3-carboxylic acid
methyl(quinolin-4-ylmethyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
5-[3-(propan-2-yloxy)phenyl]-1,2-dihydropyrimidin-2-one
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[5-(propan-2-yl)pyrimidin-4-yl]-1,4-diazepan-5-one
2-methyl-N-(oxolan-3-ylmethyl)-7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
7-[(3,4-difluorophenyl)methyl]-2-(thian-4-yl)-2,7-diazaspiro[4.5]decan-6-one
(5S)-5-({[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl](pyridin-2-ylmethyl)amino}methyl)pyrrolidin-2-one
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
N-(1-methoxypropan-2-yl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-ethyl-5-methyl-N-(2-methylprop-2-en-1-yl)-6-(4-phenylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](prop-2-en-1-yl)(pyridin-3-ylmethyl)amine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-[(4-hydroxypiperidin-1-yl)methyl]piperidin-2-one
3-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine
4-(3-hydroxy-3-methylbutyl)-N-(oxan-3-ylmethyl)benzamide
1-methyl-3-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1H-indole
2-({[(3R,4R)-1-(5-chloro-2-methylbenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
N-[(5-methylfuran-2-yl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{[(4aS,7aR)-6,6-dioxo-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
2-[2-(benzenesulfonyl)ethyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[1-(2-chlorophenyl)ethyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
1-(pyridin-3-ylmethyl)-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1,4-diazepane
1-{1'-[(3-fluoro-4-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
2-[2-(1H-imidazol-1-yl)ethyl]-1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
1-(furan-2-ylmethyl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]piperidine-3-carboxamide
5-ethyl-3-({2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2-acetyl-8-(thiophen-3-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
8-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-2-(pyrrolidin-1-yl)ethan-1-one
2-{4-[(4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,3-oxazol-2-yl)methyl]piperazin-1-yl}pyrimidine
3-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]azetidin-3-yl}pyridine
(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
N-cyclobutyl-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
4-(5-phenyl-1,2-oxazole-3-carbonyl)-1λ6-thiomorpholine-1,1-dione
N-{[8-(5-acetyl-4-methylpyrimidin-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
7-fluoro-N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-methylquinoline-4-carboxamide
3-[2-(4-ethoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2,6-dimethyl-4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}quinoline
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-3-yl]methanol
4-[3-(1,2-oxazolidine-2-carbonyl)phenoxy]-1-(2-phenylethyl)piperidine
4-[1-(1H-1,2,3-benzotriazol-5-yl)-1H-imidazol-2-yl]-N-methylbenzene-1-sulfonamide
2-{4-[1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine