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N-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
(2S,4R)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
2-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-cyclopentyl-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
4-[3-(2-chlorophenyl)-3-phenylpropanoyl]piperazin-2-one
1-(4-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
1-{1'-[2-(3-fluorophenyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
2-{4-[(3-ethyl-3-hydroxypiperidin-1-yl)methyl]phenoxy}-1-(morpholin-4-yl)ethan-1-one
N-ethyl-1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidine-3-carboxamide
2-{[4-(difluoromethoxy)phenyl]methyl}-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
{1-[({[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl)amino)methyl]cyclopentyl}methanol
(3S,4R)-1-(2-cyclopropylpyrimidine-5-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-{[5-(3-methoxyphenyl)-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4-cyclopentyl-N-{[5-(4-fluorophenyl)-1,2-oxazol-3-yl]methyl}pyrimidin-2-amine
(3R,4R)-4-cyclobutyl-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-methylpiperidin-4-ol
N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
4-[4-(1H-1,2,4-triazol-1-yl)phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(2-methoxy-4-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
3-{4-[3-(1-methylpiperidin-3-yl)propanoyl]piperazin-1-yl}benzoic acid
4-(2-phenylmorpholin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
(4aS,7aR)-N-ethyl-6,6-dioxo-4-[(1-propyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2,6-dimethyl-4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}quinoline
3-[2-(morpholin-4-yl)ethyl]-1-{4-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}urea
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylbenzamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N,5-dimethyl-N-(2-phenylethyl)thieno[2,3-d]pyrimidine-6-carboxamide
3-[4-(2-chlorophenyl)-2-methyl-5-oxopiperazine-1-carbonyl]benzonitrile
1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]isoquinoline
methyl (2R,4S)-4-hydroxy-1-[(2-methoxyquinolin-3-yl)methyl]piperidine-2-carboxylate
2-[2-({1-[4-(3-fluorophenyl)phenyl]piperidin-4-yl}amino)ethyl]-6-methyl-3,4-dihydropyrimidin-4-one
3-(2-methoxyphenyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]benzamide
(2S)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3,3-dimethylbutanamide
2-[(4aR,7aS)-4-(2-ethoxyacetyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
6-amino-2-[2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]pyrimidin-4-ol
(1S,5R)-6-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
8-[3-cyclopropyl-5-(1,4-dioxan-2-yl)-1H-1,2,4-triazol-1-yl]quinoline
9-[4-(1H-pyrazol-4-yl)butanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S,4R)-1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
2-methyl-5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidine
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(4-hydroxyphenyl)-2-phenylpropan-1-one
N-(dimethyl-1H-1,2,4-triazol-3-yl)-3-(trifluoromethyl)piperidine-1-carboxamide
5-cyclopropyl-N-[3-(pyridin-4-yl)propyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
methyl 3-cyclohexaneamido-5-{[(2-methoxyphenyl)formamido]methyl}benzoate
2-[2-(benzyloxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
benzyl 3-[2-(azocan-1-yl)-2-oxoethyl]morpholine-4-carboxylate
3-cyclohexyl-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-pyrazole-4-carboxamide
1-(3-methoxyphenyl)-4-(5-phenyl-1,2-oxazole-3-carbonyl)piperazin-2-one
1-[2-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-2-oxoethyl]pyrrolidin-2-one
2-butyl-8-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4R)-N-[(2-ethoxyphenyl)methyl]-4-hydroxy-N-(prop-2-en-1-yl)pyrrolidine-2-carboxamide
methyl 3-(2-methylbutanamido)-5-{[(3-methylthiophen-2-yl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate