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2-methyl-6-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-4H-pyran-4-one
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-(2,2-dimethyloxan-4-yl)-5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-[3-({[(4-fluorophenyl)methyl](prop-2-en-1-yl)amino}methyl)phenoxy]ethan-1-ol
1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-phenylethane-1,2-dione
5-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{3-[(2,4-difluorophenyl)methyl]-1-(6-methylquinoline-4-carbonyl)piperidin-3-yl}methanol
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]piperidine-1-sulfonamide
3-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
4-benzyl-1-(4,6-dimethylpyridine-3-carbonyl)-3-ethyl-1,4-diazepan-5-one
N-cyclohexyl-1-methyl-3-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
2-(2,5-dimethoxyphenyl)-5-methyl-4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1,3-oxazole
1-ethyl-4-{[methyl(2-phenylpropyl)amino]methyl}pyrrolidin-2-one
3-(4-hydroxyphenyl)-N-(2-methoxyethyl)-N-(oxolan-2-ylmethyl)benzamide
2-acetamido-N-[(4-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]acetamide
1-(4-{4-[2-(2-hydroxyethoxy)ethyl]piperazine-1-carbonyl}thiophen-2-yl)ethan-1-one
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-phenylpyrimidine
3-(3-methylphenyl)-1-(thiophene-3-carbonyl)piperidine
(3R,4R)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-ol
methyl 3-(1-benzofuran-2-ylmethyl)-7-oxo-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-benzyl-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
1-(methoxymethyl)-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)cyclobutane-1-carboxamide
1-(1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}cyclopentyl)pyrrolidine
[(2-ethylpyrimidin-4-yl)methyl](methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
1-[(2-fluorophenyl)methyl]-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-[5-(dimethylamino)-2-methylphenyl]-1-ethyl-1-(oxan-4-ylmethyl)urea
(2R)-1-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-2-methylpiperazine
(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
3-{[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
(4aS,7aR)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,7-dimethyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidine-5-carboxamide
3-(2-{6-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)-4-(3-methylbut-2-en-1-yl)piperazin-2-one
3-(1H-1,2,3-benzotriazol-1-yl)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethylpropanamide
1-(2-chlorophenyl)-3-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
7-cyclopentyl-2-[2-(methylamino)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-1-(piperidin-1-yl)cyclohexane-1-carboxamide
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(3,4,5-trimethoxyphenyl)methyl]piperidine
8-[(2-chloro-4-hydroxyphenyl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
2-(1-ethylpiperidin-4-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-(propan-2-yl)-7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(3-methylphenoxy)piperidine
2-methyl-8-{5-[(phenylsulfanyl)methyl]furan-2-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[2-(morpholin-4-yl)ethyl]piperidine-3,5-dicarboxamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
2-{1-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1H-imidazol-2-yl}quinoline
1-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]piperidine-4-carboxamide
2-(ethylsulfanyl)-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}propan-1-one
N-cyclobutyl-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
2-amino-4-(1,3-dimethyl-1H-pyrazol-4-yl)-6-(2-methylpropanoyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(3-chlorophenyl)-4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1H-pyrazole