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2-[2-(1H-imidazol-4-yl)ethyl]-9-(2-methyl-1,3-thiazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-fluorophenyl)methyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-[3-(propan-2-yloxy)phenyl]isoquinoline
4-{[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-({1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-1-oxopropan-2-yl}sulfanyl)-6-methyl-3,4-dihydropyrimidin-4-one
6-oxo-N-(3-phenylpropyl)piperazine-2-carboxamide
3-[(4-fluorophenyl)methyl]-1-(1H-1,2,3-triazole-5-carbonyl)piperidine
N,N-dimethyl-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]azepan-4-amine
1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-(4H-1,2,4-triazol-4-yl)benzamide
9-hydroxy-3-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
N,5-dimethyl-4-[(oxolan-2-ylmethyl)amino]-N-(thiophen-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
1-phenyl-4-({[4-(pyridin-2-yl)phenyl]methyl}amino)pyrrolidin-2-one
1-[3-(dimethylsulfamoyl)propyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
1-methyl-N-[(2S)-oxolan-2-ylmethyl]-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
3-({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)-N-(2-methoxyphenyl)propanamide
8-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(1-methyl-1H-indole-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-(cyclohex-1-en-1-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(3,5-dichloro-4-methylbenzoyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(1H-pyrazol-1-yl)butan-1-one
N-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
1-[(2-chlorophenyl)methyl]-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
3,5-dimethyl-1-{1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]azetidin-3-yl}-1H-pyrazole
3-(4-hydroxyphenyl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}benzamide
3-{1-[1-(1-acetylpiperidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-chlorophenyl)urea
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-N-(pyridin-2-ylmethyl)cyclopropanamine
4-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyrrolidin-2-one
methyl 6-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-phenyl-1,4-diazepane
4-[1-(ethanesulfonyl)piperidin-3-yl]benzoic acid
3-{2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1-phenylpiperazin-2-one
(2S,4R)-4-[(adamantan-2-yl)amino]-N-[2-(2-fluorophenyl)ethyl]-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-hydroxypropan-1-one
7-(3-chlorophenyl)-4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}({1-[2-(1H-pyrazol-1-yl)phenyl]ethyl})amine
4-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
(3R,4R)-3,4-dimethyl-1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]pyrrolidin-3-ol
1-(8-methylquinolin-5-yl)-3-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}urea
1-methyl-4-[(3-{[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-1,4-diazepane
N-benzyl-4-oxo-1-(propan-2-yl)-5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1,4-dihydropyridine-3-carboxamide
3-[(1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]propanoic acid
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-[(1-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
2-(5-ethyl-1-benzofuran-3-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
(3S,4R)-1-[2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one