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N-[(1R,3R)-3-aminocyclopentyl]-5-methoxy-3-methyl-1H-indole-2-carboxamide
3-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1-{2-[2-(pyridin-2-yl)ethyl]phenyl}urea
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(2-propoxyethyl)piperazin-1-yl]ethan-1-one
6-(4-{[2-(4-hydroxyphenyl)ethyl]amino}piperidin-1-yl)pyridine-3-carbonitrile
5-chloro-2-methoxy-4-[1-methyl-5-(piperidin-1-yl)-1H-1,2,4-triazol-3-yl]pyridine
3-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-N-(1-methyl-1H-1,3-benzodiazol-2-yl)benzamide
(2S,4R)-1-benzyl-N,N-diethyl-4-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-{3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]phenoxy}-1-(piperidin-1-yl)ethan-1-one
8-methyl-3-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-2-(thiophen-2-yl)quinoline
1-(2-methylpyridin-4-yl)-4-(6-methylpyridine-2-carbonyl)-1,4-diazepane
1-(7-methoxy-4-methylquinazolin-2-yl)-N-methyl-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]-1-(piperidin-1-yl)propan-1-one
2-methyl-N-(2-methylpropyl)-3-{[(pyrimidin-4-ylmethyl)carbamoyl]amino}benzamide
2-{5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-phenyl-1H-1,2,4-triazol-3-yl}acetamide
3-{[1-(1-methylpiperidin-4-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
[1-(1-cyclobutanecarbonylpiperidin-4-yl)-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
2-(3-ethyl-1H-indole-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(thiophen-2-yl)butanamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-5-(methoxymethyl)-N-(pyridin-4-ylmethyl)furan-2-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-1-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]propan-1-one
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-3-(N-methylmethanesulfonamido)propanamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(1H-1,2,4-triazol-3-yl)benzamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(3-phenylpiperidin-1-yl)acetamide
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-(4-methylphenoxymethyl)piperidine
ethyl 2-{[(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)carbamoyl]amino}acetate
1-(4-fluorophenyl)-6,6-dimethyl-N-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-[(3S)-3-acetamidopyrrolidin-1-yl]pyridine-2-carboxamide
N-methyl-N-(pyrazin-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-[(2-fluorophenyl)methyl]-N-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-amine
1-(pyrrolidine-1-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
4-[4-(1-methoxyethyl)phenyl]-2-methylquinazoline
3-(2-methyl-1H-imidazol-1-yl)-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]propan-1-one
4-{[4-(2-methoxybenzoyl)piperazin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
(2S)-2-{[(4-chloro-2-ethylphenyl)carbamoyl]amino}-4-methylpentanamide
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(2-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1H-indazole-3-carboxamide
1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperazine-2-carboxylic acid
(1S,5R)-3-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-({[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}amino)piperidin-1-yl]ethan-1-one
N-(2,4-dimethylphenyl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-(thiophen-3-ylmethyl)piperidine-3-carboxamide
1-cyclohexyl-4-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
5-ethyl-2-[4-(2-methylpyridin-4-yl)piperazin-1-yl]pyrimidine
ethyl 4-({[1-(pyrazin-2-yl)piperidin-3-yl]carbamoyl}amino)benzoate
6-{[2-(carbamoylmethyl)piperidin-1-yl]methyl}pyridine-2-carboxylic acid
(1R,6S)-9-methyl-N-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
(3aR,6aR)-2-{[2-(2-hydroxyethoxy)phenyl]methyl}-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3,3-diphenylpropyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(3-methylpyridin-2-yl)piperazine