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1-(4-methoxy-2-methylbenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
(3aS,7aR)-2-[2-(3-chloro-4-fluorophenyl)acetyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-{3-[(2-fluorophenyl)methoxy]azetidin-1-yl}-3-(1-methylpiperidin-2-yl)propan-1-one
1-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-N'-(3-methylphenyl)propanediamide
4-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-amido]-N-ethylpiperidine-1-carboxamide
3-(hydroxymethyl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-ol
5-(2,3-dihydro-1H-inden-2-yl)-3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-benzyl-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-3,6-diazabicyclo[3.2.2]nonane
2-(4-{[2-(methylcarbamoyl)piperidin-1-yl]methyl}phenoxy)acetic acid
N-cyclopropyl-3-(5-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanamide
(3S,4S)-1-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)-4-propylpyrrolidine-3-carboxylic acid
2-{1-[(4-fluorophenyl)methyl]-4-(quinoxalin-5-ylmethyl)piperazin-2-yl}ethan-1-ol
1-(naphthalen-1-ylmethyl)-3-(pyrrolidin-1-yl)piperidine
1-{2-[(2,5-dimethoxyphenyl)formamido]ethyl}-N-(thiophen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-{[3-(3-ethyl-4-methylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methyl}morpholine
6-chloro-3-[(3-{[(dimethylsulfamoyl)amino]methyl}piperidin-1-yl)methyl]-4H-chromen-4-one
3-({[(2-methoxyphenyl)methyl](propyl)amino}methyl)benzonitrile
1-cyclohexyl-3-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]urea
2-{3-chloro-4-[(4-fluorophenyl)methoxy]phenyl}-N,N-dimethylpyridine-3-carboxamide
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
1-[3-({4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]ethan-1-one
(furan-2-ylmethyl)({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})(thiophen-2-ylmethyl)amine
{3-[(dimethylamino)methyl]-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}methanol
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
(1R,3S,5S)-8-(6-methoxypyrimidin-4-yl)-8-azabicyclo[3.2.1]octan-3-ol
2-{[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-4-methyl-6-(trifluoromethyl)pyrimidine
N-[(3S,4R)-1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
methyl({4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl})(thiophen-3-ylmethyl)amine
2-benzyl-8-(3-ethoxypropanoyl)-2,8-diazaspiro[4.5]decan-3-one
(1R,3S)-3-(2-hydroxyethoxy)-7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-7-azaspiro[3.5]nonan-1-ol
4-methyl-2-{[2-(2-propylpyrimidin-5-yl)-1H-imidazol-1-yl]methyl}-6-(trifluoromethyl)pyrimidine
N-[1-(2-fluorophenyl)piperidin-4-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-(2H-1,3-benzodioxol-5-yl)-1-(2-methoxyphenyl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
2-[2-(4-fluorophenyl)ethyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[(3,4-dimethoxyphenyl)methyl]-4-{4-[4-(2-methylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N1-{1-[3-(4-fluorophenyl)phenyl]piperidin-4-yl}propane-1,3-diamine
2-benzyl-3-methyl-4-[2-(propan-2-yl)pyrimidin-4-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
9-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-({5-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-[(3-methyl-1-benzofuran-2-yl)methyl]-1-[2-(morpholin-4-ylmethyl)phenyl]urea
2-{2-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-1,3-thiazole-4-carboxamide
3-({2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}sulfonyl)-N,N-dimethylbenzamide
2-{[4-(2-methoxy-5-methylphenyl)-5-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-ethylbutan-1-one
N-benzyl-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
7-[2-(trifluoromethyl)morpholine-4-carbonyl]quinolin-8-ol
1-(pyridin-4-ylmethyl)-4-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]pyrrolidin-2-one
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-(1,2-oxazolidin-2-yl)propan-1-one