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4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(1,2,4-oxadiazol-3-yl)piperidine
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(quinoxalin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-chloro-4,6-dimethyl-3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,2-dihydropyridin-2-one
5-cyclopropanecarbonyl-1'-[(4-methoxy-3-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,4-diazepan-5-one
3-{[1-(4-methyl-1H-imidazole-5-carbonyl)pyrrolidin-3-yl]methyl}benzamide
N-methyl-5-propyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,2-oxazole-4-carboxamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}-4-[(4-phenylphenyl)methyl]piperazin-2-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-2-[4-(4-fluorophenyl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]acetamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(benzyloxy)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-(cyclopropylmethyl)-7-(5-phenyl-1,2-oxazole-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(3,5-dimethylphenyl)-3-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-3-oxopropanamide
5-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]pyrrolidin-2-yl}-3-phenyl-1,2,4-oxadiazole
N-(1,4-dioxan-2-ylmethyl)-4-(4-methylphenyl)-5-(pyridin-4-yl)pyrimidin-2-amine
4-{[(1R,5S)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1H-pyrazole-3-carboxylic acid
(1R,3S)-3-methoxy-7-(2-methyl-1-benzofuran-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl][2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
1-[(4-methylphenyl)methyl]-4-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}piperazin-2-one
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[2-(oxan-2-yl)ethyl]amine
2-methoxy-5-{4-phenyl-1-[3-(pyrrolidin-1-yl)propyl]-1H-imidazol-5-yl}pyrimidine
methyl 2-(ethylsulfamoyl)-6-(naphthalen-1-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{2-[({4-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)amino]ethyl}acetamide
2,4-dimethyl-6-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]pyrimidine
4-{[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
2-cyclohexyl-5-({2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidine
N-(1-cyclopentanecarbonylpiperidin-4-yl)-2-(dimethylamino)-2-(4-methylphenyl)acetamide
2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]ethan-1-one
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
N-[3-(azepan-1-yl)propyl]-3-(3-fluorophenyl)-N-methyl-1H-pyrazole-4-carboxamide
N-({3-methyl-7-[3-(prop-2-en-1-yloxy)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)methanesulfonamide
(4aR,7aS)-1-(pyridin-4-ylmethyl)-4-(pyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2-chlorophenyl)methyl]-3-methyl-4-oxo-N-(propan-2-yl)pentanamide
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-[3-benzyl-1-(4-chlorophenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
N-{1-[4-(8-methoxy-2-methylquinolin-5-yl)phenyl]ethyl}acetamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-3-amine
2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N,N-dimethylacetamide
2,3-dimethyl-6-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]quinoxaline
1-(2-methoxyphenyl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
2-hydroxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-2-[4-(trifluoromethyl)phenyl]acetamide
N-[(1S,3S)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}cyclopentyl]-1,3-thiazole-4-carboxamide
1-ethyl-5-[3-(1H-indol-3-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-({2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazol-4-yl}formamido)-N,2-dimethylpropanamide
(3S,4S)-1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-3,4-diol
1-phenyl-4-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}piperazin-2-one
1-(4-fluorophenyl)-4-[1-(pentan-3-yl)piperidin-3-yl]piperazine