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2-[1-(propan-2-yl)-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
(3aR,6aR)-2-benzoyl-5-cyclopentanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
4-[(2S)-3-hydroxy-2-methylpropyl]-1-(2-phenylphenyl)piperazin-2-one
N-benzyl-N-methyl-3-({[(2-methylpyrimidin-5-yl)methyl]amino}methyl)pyridin-2-amine
N-[2-(pyrazin-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
N-(1,3-benzoxazol-2-ylmethyl)-5,6-dimethylpyrimidin-4-amine
N-[(4-fluorophenyl)methyl]-2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
2-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-6-methylpyridine-3-carbonitrile
(1R,5S)-6-methyl-3-{2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopentyl-2-(4-oxo-3,4-dihydrophthalazin-1-yl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)propanamide
(1R,5R)-N,N-dimethyl-6-{[2-(methylsulfanyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
methyl 2-[1-(2,6-dimethylquinoline-3-carbonyl)-3-oxopiperazin-2-yl]acetate
(3S,4S)-1-[(2-chloro-6-fluorophenyl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[(3,4,5-trifluorophenyl)methyl]-1H-pyrazole-4-carboxamide
(2R,6R)-1-[2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
2-(4-{3-[(4-aminopiperidin-1-yl)methyl]-7-methylquinolin-2-yl}piperazin-1-yl)ethan-1-ol
(3S,5R)-1-(2-methoxybenzoyl)-5-(4-methylpiperazine-1-carbonyl)piperidine-3-carboxylic acid
N,N-dimethyl-5-{[(2-methylphenyl)methyl]amino}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[(2,3-difluorophenyl)methyl]-1H-pyrazole-4-carboxamide
5-methyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1-propyl-1H-pyrazole-4-carboxamide
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(3S)-2-oxoazepan-3-yl]acetamide
2-{5-[2-(2-oxoazepan-1-yl)ethyl]-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl}acetic acid
2-(2-methoxyphenyl)-8-methyl-5-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-(2H-1,3-benzodioxol-5-yl)-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]ethan-1-one
[(dimethyl-1,3-thiazol-5-yl)methyl](methyl)[2-(morpholin-4-yl)ethyl]amine
2-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1H-imidazol-2-yl}pyridine
(1R,7S)-N-(1H-imidazol-2-ylmethyl)-N-methyl-3-(3-methylbutyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-(pyrrolidine-1-carbonyl)-2-(2,3,4-trimethoxyphenyl)pyridine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[1-(1H-pyrazol-1-yl)propan-2-yl]benzamide
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-[(1-ethyl-1H-indol-3-yl)sulfanyl]ethan-1-one
4-(5,6-dimethylpyrimidin-4-yl)-2-[2-(2-methoxyethyl)-2H-1,2,3,4-tetrazol-5-yl]morpholine
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
4-benzyl-1-(5,6-dimethylpyrimidin-4-yl)-3-ethyl-1,4-diazepan-5-one
N-cyclopropyl-5-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(1-benzylpyrrolidin-3-yl)-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-(2-chlorophenyl)-3-methyl-N-(2-methylpropyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-2-[2-(thiophen-2-yl)ethyl]piperidine
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-3-(2-methyl-1H-indol-1-yl)propan-1-one
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1,3-thiazole-5-carboxamide
3-{3-[(dimethylamino)methyl]-1,2,4-oxadiazol-5-yl}-5-ethyladamantan-1-ol
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N-(2-methoxyethyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
5-(1,2-oxazol-5-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}furan-2-sulfonamide
2-(4-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}morpholin-3-yl)-N-phenylacetamide
(2E)-3-(furan-2-yl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylprop-2-enamide
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide