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5-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-[(6-chloropyridin-3-yl)methyl]-2-(2,4-dioxo-1,3-diazinan-1-yl)benzamide
5-{1H-pyrrolo[2,3-b]pyridin-1-ylmethyl}-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]urea
N-[2-(3,4-dimethoxyphenyl)ethyl]-2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N2,N2-dimethyl-N4-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
3-{[(2,2-dimethylpropyl)amino]methyl}-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
3-{1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]azetidin-3-yl}pyridine
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
4-[4-(1,3-benzothiazol-2-yl)-1,4-diazepane-1-carbonyl]-6-methylpyrimidin-2-amine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
3-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]piperidine-1-carboxamide
N-[(1R)-1-(4-methoxyphenyl)ethyl]-6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(3S,4S)-4-cyclopropyl-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]pyrrolidine-3-carboxylic acid
2-(dimethylamino)-4-methyl-N-[3-(methylsulfanyl)propyl]pyrimidine-5-carboxamide
N-{1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-methyl-1-oxobutan-2-yl}acetamide
N-cyclobutyl-5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
(2S,4R)-4-amino-1-(3-chlorothiophene-2-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(2R,3S,6R)-3-(4-methylphenyl)-5-(5-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[1-(3-methylbutyl)-5-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
2-{8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-5-propyl-1,3,4-oxadiazole
4-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]carbamoyl}amino)-3-methyl-N-(propan-2-yl)benzamide
N-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-methyl-2-(3-methylbenzoyl)-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}acetamide
diethyl({3-[2-(trifluoromethyl)morpholine-4-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
N-[2-(4-fluorophenyl)ethyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(2-ethyl-2,5-dihydro-1H-pyrrol-1-yl)sulfonyl]-N-(1-methylpiperidin-4-yl)benzamide
3-(thiophen-3-ylmethyl)-5-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,2,4-oxadiazole
2-[methyl({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl})amino]ethan-1-ol
3-fluoro-N-(1-hydroxybutan-2-yl)-7-methyl-N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
4-[1-(oxan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]quinoline
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-1,3-thiazole-5-carboxamide
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl][(4-fluorophenyl)methyl](prop-2-en-1-yl)amine
4-[1-(3-acetamidopropanoyl)piperidin-3-yl]benzoic acid
1-cyclopropyl-4-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]pyrrolidin-2-one
2-[(cyclopropylmethyl)sulfanyl]-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]ethan-1-one
3-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3,4-dihydropteridin-4-one
N-butyl-7-methoxy-N-(pyridin-4-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[(2-hydroxypropyl)sulfamoyl]-N-[3-(pyridin-4-yl)propyl]benzamide
8-(5-carboxy-1-methyl-1H-1,3-benzodiazol-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(2S,4S)-N-ethyl-1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-4-(1-methylcyclopropaneamido)pyrrolidine-2-carboxamide
(3aR,6aR)-N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
5-methyl-2-(4-{[3-(pyridine-3-carbonyl)piperidin-1-yl]methyl}piperidin-4-yl)pyridine
7-chloro-4-(4-methyl-1,3-oxazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-cyclopropylacetamide
3-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-yl)-1,3-oxazolidin-2-one
4-[(2R)-3-methylbutan-2-yl]-3-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{imidazo[1,2-a]pyridin-3-ylmethyl}(methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
N-ethyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]butanamide